SCHEMBL337602

SCHEMBL337602

Cc1cc(F)ccc1-c1cc(Cl)ncc1N

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.47
ABL1 P00519 2/20 0.39
TLR8 Q9NR97 1/20 0.35
DHFR P00374 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
UHRF1 Q96T88 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
GRM5 P41594 2/20 0.34
AGPAT2 O15120 1/20 0.33
KCNH2 Q12809 1/20 0.33
GRM2 Q14416 1/20 0.33
HSP90AB1 P08238 1/20 0.33
MAPK14 Q16539 1/20 0.33
HSD11B1 P28845 1/20 0.33
HASPIN Q8TF76 1/20 0.33
POLQ O75417 1/20 0.33
KCNA5 P22460 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30092912 1.00 GPBAR1 (0.47) GPBAR1ABL1TLR8DHFRGRIN1
SCHEMBL31756885 1.00 GPBAR1 (0.47) GPBAR1ABL1TLR8DHFRGRIN1
Hydrochloric Acid SCHEMBL28810216 0.98 GPBAR1 (0.46) GPBAR1ABL1TLR8DHFRGRIN1
SCHEMBL14600981 0.85 GPBAR1 (0.50) GPBAR1ABL1DHFRGRIN1GRIN2B
SCHEMBL1872305 0.81 GPBAR1 (0.45) GPBAR1ABL1TLR8GRIN1GRIN2B
SCHEMBL1872308 0.79 GPBAR1 (0.46) GPBAR1ABL1GRIN1GRIN2BPDE3B
SCHEMBL27729990 0.79 DPP4 (0.34) GPBAR1ABL1GRM5
SCHEMBL5783181 0.78 GPBAR1 (0.53) GPBAR1ABL1DHFRPOLQ
SCHEMBL23361562 0.76 GPBAR1 (0.46) GPBAR1GRIN1GRIN2BHSD11B1
SCHEMBL30980994 0.76 GPBAR1 (0.46) GPBAR1GRIN1GRIN2BHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12473260-B2 Chemical process for making 6-chloro-4-(4-fluoro-2-methylphenyl)pyridin-3-amine a key intermediate of NT-814 KaNDy Therapeutics Limited (GB) 2025-11-18 US claimed
US-20230002322-A1 NEW CHEMICAL PROCESS FOR MAKING 6-CHLORO-4-(4-FLUORO-2-METHYLPHENYL)PYRIDIN-3-AMINE A KEY INTERMEDIATE OF NT-814 KaNDy Therapeutics Limited (GB) 2023-01-05 US claimed
CN-114728906-A Novel chemical method for preparing key intermediate 6-chloro-4- (4-fluoro-2-methylphenyl) pyridine-3-amine of NT-814 康堤医疗有限公司 2022-07-08 CN claimed
WO-2021094247-A1 NEW CHEMICAL PROCESS FOR MAKING 6-CHLORO-4-(4-FLUORO-2-METHYLPHENYL)PYRIDIN-3-AMINE A KEY INTERMEDIATE OF NT-814 KaNDy Therapeutics Limited (GB) 2021-05-20 WO claimed
US-12473260-B2 Chemical process for making 6-chloro-4-(4-fluoro-2-methylphenyl)pyridin-3-amine a key intermediate of NT-814 KaNDy Therapeutics Limited (GB) 2025-11-18 US disclosed
US-12473260-B2 Chemical process for making 6-chloro-4-(4-fluoro-2-methylphenyl)pyridin-3-amine a key intermediate of NT-814 KaNDy Therapeutics Limited (GB) 2025-11-18 US disclosed
US-20230002322-A1 NEW CHEMICAL PROCESS FOR MAKING 6-CHLORO-4-(4-FLUORO-2-METHYLPHENYL)PYRIDIN-3-AMINE A KEY INTERMEDIATE OF NT-814 KaNDy Therapeutics Limited (GB) 2023-01-05 US disclosed
US-20230002322-A1 NEW CHEMICAL PROCESS FOR MAKING 6-CHLORO-4-(4-FLUORO-2-METHYLPHENYL)PYRIDIN-3-AMINE A KEY INTERMEDIATE OF NT-814 KaNDy Therapeutics Limited (GB) 2023-01-05 US disclosed
US-20230002322-A1 NEW CHEMICAL PROCESS FOR MAKING 6-CHLORO-4-(4-FLUORO-2-METHYLPHENYL)PYRIDIN-3-AMINE A KEY INTERMEDIATE OF NT-814 KaNDy Therapeutics Limited (GB) 2023-01-05 US disclosed
EP-4058433-A1 NEW CHEMICAL PROCESS FOR MAKING 6-CHLORO-4-(4-FLUORO-2-METHYLPHENYL)PYRIDIN-3-AMINE A KEY INTERMEDIATE OF NT-814 KaNDy Therapeutics Limited (GB) 2022-09-21 EP disclosed
CN-114728906-A Novel chemical method for preparing key intermediate 6-chloro-4- (4-fluoro-2-methylphenyl) pyridine-3-amine of NT-814 康堤医疗有限公司 2022-07-08 CN disclosed
CN-114728906-A Novel chemical method for preparing key intermediate 6-chloro-4- (4-fluoro-2-methylphenyl) pyridine-3-amine of NT-814 康堤医疗有限公司 2022-07-08 CN disclosed
US-20110190276-A1 Pyridine Derivatives And Their Use In The Treatment Of Psychotic Disorders KaNDy Therapeutics Limited (GB) 2011-08-04 US disclosed
EP-2336136-A1 Pyridine derivatives and their use in the treatment of psychotic disorders GlaxoSmithKline LLC (US) 2011-06-22 EP disclosed
US-7919491-B2 Pyridine derivatives and their use in the treatment of psychotic disorders GLAXOSMITHKLINE LLC (US) 2011-04-05 US disclosed
US-20100152175-A1 Pyridine Derivatives and Their Use in The Treatment of Psychotic Disorders GLAXOSMITHKLINE LLC (US) 2010-06-17 US disclosed
US-7683056-B2 Pyridine derivatives and their use in the treatment of psychotic disorders GLAXOSMITHKLINE LLC (US) 2010-03-23 US disclosed
US-20080269208-A1 Pyridine Derivatives and Their Use in the Treatment of Psychotic Disorders KaNDy Therapeutics Limited (GB) 2008-10-30 US disclosed
EP-1928886-A1 PYRIDINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF PSYCHOTIC DISORDERS SmithKline Beecham Corporation (US) 2008-06-11 EP disclosed
WO-2007028654-A1 PYRIDINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF PSYCHOTIC DISORDERS SMITHKLINE BEECHAM CORPORATION (US) 2007-03-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110190276-A1 Pyridine Derivatives And Their Use In The Treatment Of Psychotic Disorders NDUFB7, NDUFB6, GABRE GPBAR1 1351/4885ABL1 574/4885TLR8 2879/4885
US-20230002322-A1 NEW CHEMICAL PROCESS FOR MAKING 6-CHLORO-4-(4-FLUORO-2-METHYLPHENYL)PYRIDIN-3-AMINE A KEY INTERMEDIATE OF NT-814 NT5E, NT5M, NTRK2 GPBAR1 3570/4885ABL1 332/4885TLR8 1596/4885
US-20080269208-A1 Pyridine Derivatives and Their Use in the Treatment of Psychotic Disorders SLC6A3, NDUFS5, NDUFB6 GPBAR1 1490/4885ABL1 109/4885TLR8 2838/4885
US-20100152175-A1 Pyridine Derivatives and Their Use in The Treatment of Psychotic Disorders CHRNA7, NR3C2, CHRNA6 GPBAR1 783/4885ABL1 600/4885TLR8 2057/4885
US-12473260-B2 Chemical process for making 6-chloro-4-(4-fluoro-2-methylphenyl)pyridin-3-amine a key intermediate of NT-814 NT5E, NT5M, NTRK2 GPBAR1 3309/4885ABL1 242/4885TLR8 1432/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.