SCHEMBL3379043

SCHEMBL3379043

Nc1c(C(F)(F)F)cc(Cl)c(C(F)(F)F)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 4/20 0.39
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
HTR3A P46098 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37
ADRB2 P07550 5/20 0.36
ADRB1 P08588 1/20 0.36
IDO1 P14902 2/20 0.33
GLA P06280 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
TSHR P16473 1/20 0.33
NPFFR2 Q9Y5X5 3/20 0.33
NPFFR1 Q9GZQ6 2/20 0.33
ALDH1A1 P00352 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4634857 0.83 NOTUM (0.42) NOTUMHTR3AADRB2ADRB1GAA
SCHEMBL27680544 0.76 ADRB2 (0.37) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL10616182 0.74 ALDH1A1 (0.39) NOTUMHTR3EHTR3BHTR3AHTR3D
SCHEMBL9852678 0.73 ADRB2 (0.38) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL27680558 0.73 ADRB2 (0.41) NOTUMHTR3EHTR3BHTR3AHTR3D
SCHEMBL1263100 0.73 IDO1 (0.37) NOTUMHTR3EHTR3BHTR3AHTR3D
SCHEMBL24616502 0.72 TSHR (0.43) NOTUMHTR3EHTR3BHTR3AHTR3D
SCHEMBL2957239 0.72 NOTUM (0.38) NOTUMHTR3EHTR3BHTR3AHTR3D
SCHEMBL11602314 0.71 NOTUM (0.40) NOTUMHTR3EHTR3BHTR3AHTR3D
SCHEMBL9748215 0.71 ALDH1A1 (0.36) NOTUMHTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968578-A2 POLYMORPHS AND AMORPHOUS FORMS OF 5-AMINO-l-[2,6- DICHLORO-4-(TRIFLUOROMETHYL)PHENYL]-4- [(TRIFLUOROMETHYL)SULFINYL]-IH-PYRAZOLE-3-CARBONITRILE MAKHTESHIM CHEMICAL WORKS LIMITED (IL) 2008-09-17 EP claimed
WO-2007069254-A2 POLYMORPHS AND AMORPHOUS FORMS OF 5-AMINO-l-[2,6- DICHLORO-4-(TRIFLUOROMETHYL)PHENYL]-4- [(TRIFLUOROMETHYL)SULFINYL]-IH-PYRAZOLE-3-CARBONITRILE MAKHTESHIM CHEMICAL WORKS LTD. (IL) 2007-06-21 WO claimed
WO-2010049789-A1 PROCESS FOR THE SYNTHESIS OF FIPRONIL DYNAMIT NOBEL GMBH EXPLOSIVSTOFF-UND SYSTEMTECHNICK (DE) 2010-05-06 WO disclosed