SCHEMBL3380179

SCHEMBL3380179

N#Cc1ccccc1-c1ccc(Cc2cc(-c3ccccc3)n3nccc3n2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 4/20 0.41
GABRB3 P28472 4/20 0.41
GABRA1 P14867 3/20 0.41
GABRA2 P47869 3/20 0.41
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
CYP19A1 P11511 3/20 0.39
AXL P30530 1/20 0.38
FLT3 P36888 1/20 0.38
MERTK Q12866 1/20 0.38
KDM4E B2RXH2 3/20 0.38
HPGD P15428 3/20 0.38
ALDH1A1 P00352 2/20 0.38
GLA P06280 1/20 0.38
MAPK1 P28482 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PPARG P37231 2/20 0.38
CNR2 P34972 1/20 0.37
ESR2 Q92731 1/20 0.36
GABRA5 P31644 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9262125 0.75 AXL (0.41) GABRG2GABRB3GABRA1GABRA2GSK3A
SCHEMBL7437667 0.74 PRKAB2 (0.51) GSK3BALDH1A1MAPK1HSD17B10PPARG
SCHEMBL7445604 0.74 KCNN3 (0.66) ALDH1A1MAPK1HSD17B10PPARGCLK4
SCHEMBL7438857 0.73 GSK3B (0.48) GABRG2GABRB3GABRA1GABRA2GSK3A
SCHEMBL7438169 0.73 AXL (0.47) GABRG2GABRB3GABRA1GABRA2GSK3A
SCHEMBL7320243 0.73 PPARG (0.47) GSK3AGSK3BAXLFLT3MERTK
SCHEMBL7441417 0.72 MEN1 (0.49) ALDH1A1MAPK1HSD17B10MAPTCLK4
SCHEMBL9262231 0.71 PPARG (0.46) GSK3AGSK3BAXLFLT3MERTK
SCHEMBL7435705 0.71 KCNN3 (0.46) PPARG
SCHEMBL30904901 0.71 KDM4E (0.44) KDM4EHPGDALDH1A1GLAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059838-A2 PDE4 INHIBITORS SELECTIVE FOR THE LONG FORM OF PDE4 FOR TREATING INFLAMMATION AND AVOIDING SIDE EFFECTS DECODE GENETICS EHF (IS) 2010-05-27 WO claimed
WO-2010059836-A1 SUBSTITUTED AZA-BRIDGED BICYCLICS FOR CARDIOVASCULAR AND CNS DISEASE DECODE GENETICS EHF (IS) 2010-05-27 WO claimed