SCHEMBL3381301

SCHEMBL3381301

CC(Cc1ccc(-c2ccn3c(-c4ccc(CC(=O)Nc5cc(C(C)(C)C)ccn5)c(F)c4)cnc3c2)cn1)N1CCOCC1

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDR P35968 11/20 0.35
FGFR3 P22607 11/20 0.35
SIK2 Q9H0K1 2/20 0.34
SIK3 Q9Y2K2 2/20 0.34
SIK1 P57059 1/20 0.34
KIT P10721 2/20 0.34
CTSC P53634 1/20 0.33
NTRK1 P04629 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3186140 0.95 FGFR3 (0.36) KDRFGFR3SIK2SIK3SIK1
SCHEMBL3186146 0.95 FGFR3 (0.36) KDRFGFR3SIK2SIK3SIK1
SCHEMBL3384199 0.91 FGFR3 (0.39) KDRFGFR3
SCHEMBL3188986 0.90 RIPK3 (0.38) KDRFGFR3SIK2SIK3SIK1
SCHEMBL3383420 0.89 KDR (0.36) KDRFGFR3CTSCNTRK1
SCHEMBL3385611 0.85 KDR (0.36) KDRFGFR3SIK2SIK3SIK1
SCHEMBL3196972 0.82 FGFR3 (0.35) KDRFGFR3SIK2SIK3SIK1
SCHEMBL3196988 0.82 FGFR3 (0.35) KDRFGFR3SIK2SIK3SIK1
SCHEMBL3382504 0.81 KDR (0.47) KDRFGFR3NTRK1
SCHEMBL3386163 0.81 WNT3A (0.42) KDRFGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed