SCHEMBL3385476

SCHEMBL3385476

O=C(Cc1ccc(-c2cnc3cc(-c4ccncc4)ccn23)cc1)Nc1cc(C(F)(F)F)ccc1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 12/20 0.49
FGFR3 P22607 10/20 0.49
DDR1 Q08345 1/20 0.48
RET P07949 1/20 0.43
CSF1R P07333 2/20 0.41
FLT3 P36888 2/20 0.41
NEK2 P51955 2/20 0.41
NTRK1 P04629 2/20 0.41
PLK4 O00444 1/20 0.41
AURKA O14965 1/20 0.41
MAPK13 O15264 1/20 0.41
PDPK1 O15530 1/20 0.41
JAK2 O60674 1/20 0.41
CHEK2 O96017 1/20 0.41
ABL1 P00519 1/20 0.41
INSR P06213 1/20 0.41
LCK P06239 1/20 0.41
FYN P06241 1/20 0.41
LYN P07948 1/20 0.41
MET P08581 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3385250 0.89 FLT3 (0.47) KDRFGFR3DDR1RETCSF1R
SCHEMBL3385219 0.88 KDR (0.53) KDRFGFR3DDR1
SCHEMBL3385496 0.86 KDR (0.50) KDRFGFR3RETNTRK1GSK3B
SCHEMBL3195980 0.85 RET (0.60) KDRFGFR3DDR1RETABL1
SCHEMBL3417117 0.82 WNT3A (0.49) KDRFGFR3
SCHEMBL3381109 0.79 RET (0.56) KDRFGFR3RET
SCHEMBL3384065 0.79 KDR (0.52) KDRFGFR3CSF1RFLT1
SCHEMBL3384190 0.79 KDR (0.62) KDRFGFR3NTRK1
SCHEMBL31481233 0.79 KDR (0.47) KDRRETCSF1RPDPK1KIT
SCHEMBL3385818 0.78 KDR (0.49) KDRFGFR3DDR1ABL1KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101128461-B Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI 2010-12-22 CN disclosed
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed
CN-101128461-A Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors LILLY CO ELI (US) 2008-02-20 CN disclosed