SCHEMBL3384343

SCHEMBL3384343

Cc1cc(-c2ccn3c(-c4ccc(CC(=O)Nc5cc(C(C)(C)C)cc(CN6CCOCC6)n5)c(F)c4)cnc3c2)ccn1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
WNT3A P56704 7/20 0.39
KDR P35968 7/20 0.38
FGFR3 P22607 4/20 0.38
WNT1 P04628 2/20 0.36
GSK3B P49841 2/20 0.36
DYRK1A Q13627 2/20 0.36
MAPK13 O15264 1/20 0.35
MAPK12 P53778 1/20 0.35
MAPK11 Q15759 1/20 0.35
MAPK14 Q16539 1/20 0.35
RET P07949 1/20 0.35
BDKRB1 P46663 1/20 0.35
USP30 Q70CQ3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3202028 0.93 KDR (0.41) KDRFGFR3WNT1GSK3BDYRK1A
SCHEMBL3386227 0.90 KDR (0.43) KDRFGFR3RETBDKRB1
SCHEMBL3386163 0.85 WNT3A (0.42) WNT3AKDRFGFR3
SCHEMBL3383517 0.83 KDR (0.44) KDRFGFR3
SCHEMBL3189267 0.82 KDR (0.45) WNT3AKDRFGFR3
SCHEMBL3379613 0.82 KDR (0.37) KDRFGFR3WNT1GSK3BDYRK1A
SCHEMBL3386457 0.82 DDR1 (0.42) WNT3AKDRFGFR3RETBDKRB1
SCHEMBL3385477 0.82 FGFR3 (0.41) KDRFGFR3
SCHEMBL3186146 0.81 FGFR3 (0.36) KDRFGFR3
SCHEMBL3186140 0.81 FGFR3 (0.36) KDRFGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed