SCHEMBL3386227

SCHEMBL3386227

CC(C)(C)c1cc(CN2CCOCC2)nc(NC(=O)Cc2ccc(-c3cnc4cc(-c5ccccn5)ccn34)cc2F)c1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDR P35968 13/20 0.43
FGFR3 P22607 10/20 0.43
MOK Q9UQ07 1/20 0.38
TGFBR1 P36897 1/20 0.36
TGFBR2 P37173 1/20 0.36
RET P07949 1/20 0.36
BDKRB1 P46663 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3383517 0.94 KDR (0.44) KDRFGFR3
SCHEMBL3202028 0.91 KDR (0.41) KDRFGFR3RETBDKRB1
SCHEMBL3384343 0.90 WNT3A (0.39) KDRFGFR3RETBDKRB1
SCHEMBL3386379 0.85 FGFR3 (0.42) KDRFGFR3MOK
SCHEMBL3383240 0.84 FGFR3 (0.49) KDRFGFR3
SCHEMBL3384104 0.83 FGFR3 (0.46) KDRFGFR3RET
SCHEMBL3385167 0.81 KDR (0.39) KDRFGFR3MOKBDKRB1
SCHEMBL3189878 0.81 KDR (0.49) KDRFGFR3RET
SCHEMBL3384199 0.80 FGFR3 (0.39) KDRFGFR3
SCHEMBL3386457 0.80 DDR1 (0.42) KDRFGFR3RETBDKRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed