SCHEMBL3385140

SCHEMBL3385140

OC(c1ccc(-c2ccccc2-c2ccsc2)cc1)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.48
NR1H2 P55055 9/20 0.41
NR1H3 Q13133 9/20 0.41
TOP1 P11387 1/20 0.40
RORC P51449 3/20 0.39
RORA P35398 1/20 0.39
CYP2E1 P05181 1/20 0.39
CYP2A6 P11509 1/20 0.39
CYP2B6 P20813 1/20 0.39
PTPRC P08575 1/20 0.39
MLYCD O95822 2/20 0.38
ENPP1 P22413 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3387925 0.77 PDK2 (0.48) PDK2NR1H2NR1H3RORCRORA
SCHEMBL4946960 0.75 CYP2A6 (0.64) PDK2CYP2E1CYP2A6CYP2B6PTPRC
SCHEMBL28753042 0.75 PDK2 (0.47) PDK2NR1H2NR1H3RORCRORA
SCHEMBL28507379 0.73 NR1H2 (0.50) PDK2NR1H2NR1H3RORCRORA
SCHEMBL28930463 0.73 ALDH1A1 (0.50) NR1H2NR1H3RORCRORAMLYCD
SCHEMBL3385529 0.73 ALDH1A1 (0.50) PDK2NR1H2NR1H3RORCRORA
SCHEMBL7058734 0.73 CYP2A6 (0.70) PDK2CYP2E1CYP2A6CYP2B6PTPRC
SCHEMBL12759665 0.73 NR1H2 (0.43) NR1H2NR1H3RORCRORAMLYCD
SCHEMBL27870289 0.72 CYP2A6 (0.67) PDK2CYP2E1CYP2A6CYP2B6PTPRC
SCHEMBL19149374 0.72 NR1H3 (0.60) NR1H2NR1H3MLYCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010023317-A1 NOVEL HEXAFLUORO-2-BIPHENYLISOPROPANOL COMPOUNDS THAT MODULATE LXR-TYPE RECEPTORS, PROCESS FOR THE PREPARATION THEREOF AND USE THEREOF AS MEDICAMENTS IN HUMAN AND VETERINARY MEDICINE AND ALSO IN COSMETICS GALDERMA RESEARCH & DEVELOPMENT (FR) 2010-03-04 WO disclosed