SCHEMBL3386477

SCHEMBL3386477

CCC(C)(CC)c1cc(NC(=O)NCc2ccc(-c3cnc4cc(-c5ccncc5)ccn34)cc2)on1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDR P35968 14/20 0.47
FGFR3 P22607 12/20 0.47
MAPK13 O15264 1/20 0.39
MAPK14 Q16539 1/20 0.39
FLT3 P36888 1/20 0.39
PPID Q08752 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3385035 0.93 KDR (0.49) KDRFGFR3MAPK13MAPK14FLT3
SCHEMBL3381305 0.91 KDR (0.46) KDRFGFR3MAPK13MAPK14FLT3
SCHEMBL3383467 0.91 FLT3 (0.44) KDRFGFR3FLT3
SCHEMBL3383255 0.84 KDR (0.55) KDRFGFR3MAPK13MAPK14
SCHEMBL3383349 0.83 FLT3 (0.47) KDRFGFR3FLT3
SCHEMBL3385534 0.82 KDR (0.50) KDRFGFR3MAPK13MAPK14FLT3
SCHEMBL3386223 0.82 FLT3 (0.43) KDRFGFR3FLT3
SCHEMBL3385889 0.81 RAF1 (0.56) KDRFGFR3MAPK13MAPK14FLT3
SCHEMBL3385590 0.81 MAPK14 (0.40) KDRFGFR3MAPK13MAPK14FLT3
SCHEMBL3385883 0.79 KDR (0.50) KDRFGFR3MAPK13MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904494-B1 IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS LILLY CO ELI (US) 2010-12-01 EP disclosed