SCHEMBL3389451

SCHEMBL3389451

N#CC1(Cc2ccc(F)cc2)CCN(C(=O)c2cnn3cccnc23)CC1.N#CN1CC(C(=O)N2CCC(C#N)(Cc3ccc(F)cc3)CC2)Oc2ccc(Cl)cc21

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
ALDH1A1 P00352 1/20 0.39
KDM4E B2RXH2 1/20 0.39
NAMPT P43490 1/20 0.39
JAK2 O60674 2/20 0.38
JAK1 P23458 2/20 0.38
IRAK4 Q9NWZ3 9/20 0.37
GAA P10253 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
TSHR P16473 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3359501 0.87 ALDH1A1 (0.38) POLBALDH1A1
SCHEMBL3353428 0.82 HTR2A (0.54) POLBHTR2AHTR2CALDH1A1KDM4E
SCHEMBL13308402 0.79 ALDH1A1 (0.39) POLBALDH1A1KDM4E
SCHEMBL3355499 0.76 ALDH1A1 (0.42) POLBALDH1A1
SCHEMBL3355372 0.75 ALDH1A1 (0.35) ALDH1A1
SCHEMBL3356345 0.75 ALDH1A1 (0.37) POLBALDH1A1KDM4E
SCHEMBL3353011 0.74 LMNA (0.34) ALDH1A1KDM4E
SCHEMBL3353857 0.74 ALDH1A1 (0.36) POLBALDH1A1
SCHEMBL3359150 0.73 ADAMTS5 (0.40) ALDH1A1
SCHEMBL3353123 0.70 HTR1A (0.37) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010068881-A1 NOVEL BENZODIOXANE AND BENZOXAZINE DERIVATIVES USEFUL AS CC CHEMOKINE RECEPTOR LIGANDS FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-06-17 WO disclosed