SCHEMBL3390345

SCHEMBL3390345

CCN(CC)CCCCNc1nc(C)cc(NCCc2c[nH]c3ccc(O)cc23)n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 2/20 0.55
KDM4E B2RXH2 3/20 0.47
HTR2C P28335 2/20 0.47
CYP2D6 P10635 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
IP6K1 Q92551 1/20 0.46
SLC6A4 P31645 2/20 0.45
HTR1A P08908 1/20 0.44
HTR2A P28223 1/20 0.44
SPR P35270 3/20 0.44
ALDH1A1 P00352 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
MPO P05164 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPT P10636 1/20 0.44
IDO1 P14902 1/20 0.44
HPGD P15428 1/20 0.44
BLM P54132 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3389960 0.87 HTR1D (0.53) HTR1DKDM4EHTR2CCYP2D6MEN1
SCHEMBL3388954 0.87 HTR1D (0.53) HTR1DKDM4EHTR2CCYP2D6MEN1
SCHEMBL2599242 0.77 HTR2C (0.47) HTR1DKDM4EHTR2CCYP2D6MEN1
SCHEMBL3388179 0.76 HTR1A (0.49) MEN1KMT2AHTR1AHTR2AMAPT
SCHEMBL31379883 0.76 HTR1A (0.49) MEN1KMT2AHTR1AHTR2AMAPT
SCHEMBL23069123 0.73 HTR1D (1.00) HTR1DKDM4EHTR2CCYP2D6MEN1
SCHEMBL30276871 0.68 HTR1D (0.90) HTR1DKDM4EHTR2CCYP2D6MEN1
SCHEMBL24243759 0.68 HTR1D (0.90) HTR1DKDM4EHTR2CCYP2D6MEN1
SCHEMBL22639757 0.68 HTR2A (0.56) KDM4EMEN1KMT2AIP6K1HTR1A
SCHEMBL28152048 0.67 HTR2C (0.51) HTR1DKDM4EHTR2CCYP2D6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2241555-A1 New RAC1 inhibitors as potential pharmacological agents for heart failure treatment UNIVERSITA' DEGLI STUDI DI MILANO (IT) 2010-10-20 EP claimed
EP-2241555-A1 New RAC1 inhibitors as potential pharmacological agents for heart failure treatment UNIVERSITA' DEGLI STUDI DI MILANO (IT) 2010-10-20 EP disclosed