SCHEMBL3391740

SCHEMBL3391740

CCOc1cc(C(F)(F)F)n(-c2ccncc2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.42
EPHX2 P34913 3/20 0.36
DGAT1 O75907 1/20 0.36
PTGS2 P35354 4/20 0.35
PTGS1 P23219 2/20 0.35
PPARD Q03181 1/20 0.35
PPARA Q07869 1/20 0.35
TRPC3 Q13507 2/20 0.34
TRPC1 P48995 1/20 0.34
STIM1 Q13586 1/20 0.34
ORAI1 Q96D31 1/20 0.34
TGFBR1 P36897 1/20 0.33
KDM4E B2RXH2 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAPK14 Q16539 1/20 0.32
GAA P10253 1/20 0.32
SRC P12931 1/20 0.32
BRAF P15056 1/20 0.32
KDR P35968 1/20 0.32
SCN9A Q15858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3390256 0.87 PKM (0.46) PKMDGAT1PTGS1
SCHEMBL3390287 0.84 EPHX2 (0.40) PKMEPHX2DGAT1PPARDPPARA
SCHEMBL29864222 0.82 PKM (0.42) PKMEPHX2PTGS2PTGS1PPARD
SCHEMBL4246326 0.80 PKM (0.36) PKMEPHX2PTGS2PTGS1TRPC3
SCHEMBL4252779 0.79 PKM (0.36) PKMEPHX2PTGS2PTGS1TRPC3
SCHEMBL13495083 0.74 TGFBR1 (0.48) PTGS2PTGS1TGFBR1KDM4E
SCHEMBL4253821 0.74 KMT2A (0.43) PKMEPHX2PTGS2PTGS1GAA
SCHEMBL13702075 0.73 NPC1 (0.38) PKMEPHX2PTGS2PTGS1KDM4E
SCHEMBL27881287 0.70 PTGS1 (0.43) PKMPTGS2PTGS1
SCHEMBL17290871 0.65 BCL2 (0.46) KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2151433-A1 Alkoxypyrazoles and the process for their preparation Institut Pasteur (FR) 2010-02-10 EP disclosed
EP-2151433-A1 Alkoxypyrazoles and the process for their preparation Institut Pasteur (FR) 2010-02-10 EP disclosed