SCHEMBL3393523

SCHEMBL3393523

C=C(c1cccc(Br)c1)c1cccc(OCCl)c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAOB P27338 9/20 0.46
MRGPRX4 Q96LA9 1/20 0.43
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 1/20 0.41
MAOA P21397 1/20 0.40
GRM4 Q14833 1/20 0.40
SMPD1 P17405 1/20 0.40
TP53 P04637 1/20 0.39
AKR1C2 P52895 1/20 0.39
AKR1C1 Q04828 1/20 0.39
KMT2A Q03164 1/20 0.39
C1S P09871 1/20 0.39
PARP1 P09874 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3395887 0.84 MAOB (0.46) MAOBMRGPRX4NPC1RAB9ASMN1; SMN2
SCHEMBL2431860 0.81 MAOB (0.60) MAOBMRGPRX4RAB9AALDH1A1GRM4
SCHEMBL8865210 0.79 C1S (0.56) NPC1SMN1; SMN2ALDH1A1TP53KMT2A
SCHEMBL2278961 0.79 CES2 (0.53) MAOBNPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL2281706 0.75 RAB9A (0.45) MAOBNPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL2284121 0.75 MAOB (0.47) MAOBMRGPRX4NPC1SMN1; SMN2ALDH1A1
SCHEMBL1744811 0.74 C1S (0.50) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL12251468 0.72 LMNA (0.54) MAOBNPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL2277164 0.72 TDP1 (0.45) MAOBMRGPRX4NPC1RAB9ASMN1; SMN2
SCHEMBL2283828 0.71 CTSL (0.49) SMN1; SMN2ALDH1A1TP53KMT2AC1S

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245019-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2010-11-03 EP disclosed
WO-2009103626-A1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed