SCHEMBL3398472

SCHEMBL3398472

COc1cc(F)c(-c2nc(C)c(C(=O)N3CCN(C4CCCC4)CC3)s2)cc1F

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.44
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
HTR2C P28335 7/20 0.42
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.41
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
LRRK2 Q5S007 1/20 0.38
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13309677 0.92 HTR2C (0.46) HTR2CALDH1A1KDM4ELMNA
SCHEMBL3402527 0.92 HTR2C (0.46) HTR2CALDH1A1KDM4ELMNA
SCHEMBL3403568 0.86 RAB9A (0.45) PKMNPC1RAB9AALDH1A1HPGD
SCHEMBL3405124 0.86 NPC1 (0.45) PKMNPC1RAB9AHTR2CALDH1A1
SCHEMBL3398946 0.84 PKM (0.48) PKMNPC1RAB9AHTR2CALDH1A1
SCHEMBL3405361 0.84 RAB9A (0.53) PKMNPC1RAB9AHTR2CALDH1A1
SCHEMBL3402627 0.84 RAB9A (0.50) PKMNPC1RAB9AHTR2CALDH1A1
SCHEMBL3400125 0.83 HTR2C (0.56) PKMNPC1RAB9AHTR2CALDH1A1
SCHEMBL3404973 0.83 HTR2C (0.46) NPC1RAB9AHTR2CALDH1A1HPGD
SCHEMBL3405439 0.83 HTR2C (0.46) HTR2CALDH1A1HPGDLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed