SCHEMBL3399276

SCHEMBL3399276

COCCOC(=O)C1=C(C)N(c2ccccc2OC)C2=C(C1)C(=O)CCC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.39
KDM4E B2RXH2 4/20 0.39
ALDH1A1 P00352 3/20 0.39
HPGD P15428 3/20 0.39
GAA P10253 2/20 0.39
RUNX1 Q01196 1/20 0.39
CBFB Q13951 1/20 0.39
HKDC1 Q2TB90 1/20 0.39
TSHR P16473 2/20 0.37
CHRM5 P08912 2/20 0.36
CHRM1 P11229 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HTT P42858 1/20 0.36
RECQL P46063 1/20 0.36
KMT2A Q03164 1/20 0.36
MAPK1 P28482 1/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
BAP1 Q92560 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10722931 0.68 DRD2 (0.55) MAPTKDM4EALDH1A1CHRM5CHRM1
SCHEMBL10823922 0.65 ALDH1A1 (0.41) MAPTKDM4EALDH1A1HPGDGAA
SCHEMBL10439090 0.65 KDM4E (0.51) MAPTKDM4EALDH1A1GAATSHR
SCHEMBL3325678 0.62 ALDH1A1 (0.74) KDM4EALDH1A1HPGDGAATSHR
SCHEMBL8115164 0.58 GAA (0.63) MAPTKDM4EALDH1A1HPGDGAA
SCHEMBL317670 0.57 TSHR (0.47) KDM4EALDH1A1HPGDTSHRCHRM5
SCHEMBL29389335 0.57 TSHR (1.00) KDM4EALDH1A1HPGDTSHRSMN1; SMN2
SCHEMBL186285 0.57 TSHR (1.00) KDM4EALDH1A1HPGDTSHRSMN1; SMN2
SCHEMBL3265630 0.56 MAPT (0.64) MAPTKDM4EALDH1A1HPGDGAA
1,2-Dimethoxybenzene SCHEMBL10829425 0.56 CA1 (0.72) ALDH1A1TSHRSMN1; SMN2HTTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2249818-A1 HEDGEHOG PATHWAY ANTAGONISTS AND METHODS OF USE Stanford University (US) 2010-11-17 EP disclosed