SCHEMBL3399648

SCHEMBL3399648

O=C(NC1COCCn2c1nc(-c1ccncn1)cc2=O)c1cc(F)cc2c1OCOC2

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 1/20 0.43
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
CXCR5 P32302 1/20 0.38
GSK3B P49841 13/20 0.34
CYP1A2 P05177 6/20 0.34
CYP2D6 P10635 6/20 0.34
CSNK1A1 P48729 1/20 0.34
GSK3A P49840 1/20 0.34
F11 P03951 1/20 0.34
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
GALR3 O60755 1/20 0.32
NR2F2 P24468 1/20 0.32
USP30 Q70CQ3 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3663057 0.88 KDM4E (0.42) KDM4EALDH1A1NPC1RAB9ACXCR5
SCHEMBL3398498 0.81 GSK3B (0.38) GSK3BCYP1A2CYP2D6CNR1CNR2
SCHEMBL3399343 0.80 GSK3B (0.47) GSK3BCYP1A2CYP2D6CSNK1A1GSK3A
SCHEMBL3403548 0.79 GSK3B (0.34) GSK3BCYP1A2CYP2D6CNR1CNR2
SCHEMBL3402173 0.79 GSK3B (0.45) GSK3BCYP1A2CYP2D6
SCHEMBL3661770 0.79 KDM4E (0.44) KDM4EALDH1A1NPC1RAB9ACXCR5
SCHEMBL3401042 0.76 GSK3B (0.39) NPC1RAB9AGSK3BCYP1A2CYP2D6
SCHEMBL3400870 0.76 GSK3B (0.42) GSK3BCYP1A2CYP2D6
SCHEMBL3402193 0.76 GSK3B (0.42) GSK3BCYP1A2CYP2D6
SCHEMBL3662202 0.75 KDM4E (0.45) KDM4EALDH1A1NPC1RAB9ACXCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247598-A1 SUBSTITUTED HETEROARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2010-11-10 EP disclosed
WO-2009095787-A1 SUBSTITUTED HETEROARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2009-08-06 WO disclosed