SCHEMBL3403548

SCHEMBL3403548

Nc1c(Cl)cc(C(=O)NC2COCCn3c2nc(-c2ccncn2)cc3=O)c2c1OCCO2

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 11/20 0.34
HTR4 Q13639 3/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2D6 P10635 2/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
HTR1A P08908 1/20 0.32
ADRA2C P18825 1/20 0.32
ACHE P22303 1/20 0.32
PTGS1 P23219 1/20 0.32
ADRA1A P35348 1/20 0.32
HTR3A P46098 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3788227 0.89 GSK3B (0.42) GSK3BHTR4CYP1A2CYP2D6HTR3A
SCHEMBL3400823 0.84 HTR4 (0.42) HTR4CYP1A2CYP2D6ADRA2CACHE
SCHEMBL3398498 0.81 GSK3B (0.38) GSK3BCYP1A2CYP2D6CNR1CNR2
SCHEMBL3399684 0.79 CRBN (0.42) GSK3BCYP1A2CYP2D6
SCHEMBL927355 0.79 GSK3B (0.39) GSK3BCYP1A2CYP2D6
SCHEMBL3425658 0.79 KCNMA1 (0.40) GSK3BCYP1A2CYP2D6
SCHEMBL3399648 0.79 KDM4E (0.43) GSK3BCYP1A2CYP2D6CNR1CNR2
SCHEMBL3402173 0.78 GSK3B (0.45) GSK3BCYP1A2CYP2D6
SCHEMBL3400870 0.77 GSK3B (0.42) GSK3BCYP1A2CYP2D6
SCHEMBL3401042 0.77 GSK3B (0.39) GSK3BCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247598-A1 SUBSTITUTED HETEROARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2010-11-10 EP claimed
WO-2009095787-A1 SUBSTITUTED HETEROARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2009-08-06 WO claimed
EP-2247598-A1 SUBSTITUTED HETEROARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2010-11-10 EP disclosed
WO-2009095787-A1 SUBSTITUTED HETEROARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2009-08-06 WO disclosed