SCHEMBL3399723

SCHEMBL3399723

COc1cccc(OC)c1-c1nc(C)c(C(=O)NCCCN2CCCCC2C)s1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
TSHR P16473 1/20 0.51
CYP2C19 P33261 1/20 0.51
RAB9A P51151 2/20 0.48
NPC1 O15118 1/20 0.48
THRB P10828 1/20 0.47
SLC2A1 P11166 2/20 0.45
HRH3 Q9Y5N1 1/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPK1 P28482 1/20 0.44
CACNA1G O43497 2/20 0.44
LMNA P02545 3/20 0.43
TP53 P04637 2/20 0.43
MAPT P10636 2/20 0.43
ALDH1A1 P00352 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3399710 0.89 THRB (0.54) HSD17B10CYP1A2CYP2D6CYP2C9TSHR
SCHEMBL3399980 0.88 RAB9A (0.49) HSD17B10CYP1A2CYP2D6CYP2C9TSHR
SCHEMBL3405639 0.86 HSD17B10 (0.49) HSD17B10CYP1A2CYP2D6CYP2C9TSHR
SCHEMBL3406018 0.86 HSD17B10 (0.49) HSD17B10CYP1A2CYP2D6CYP2C9TSHR
SCHEMBL3402499 0.86 CYP1A2 (0.53) HSD17B10CYP1A2CYP2D6CYP2C9TSHR
SCHEMBL3402383 0.86 HSD17B10 (0.51) HSD17B10CYP1A2CYP2D6CYP2C9TSHR
SCHEMBL3400138 0.86 HSD17B10 (0.53) HSD17B10CYP1A2CYP2D6CYP2C9TSHR
SCHEMBL3400068 0.85 CYP1A2 (0.58) HSD17B10CYP1A2CYP2D6CYP2C9TSHR
SCHEMBL13071990 0.84 HSD17B10 (0.51) HSD17B10CYP1A2CYP2D6CYP2C9TSHR
SCHEMBL3401951 0.84 HSD17B10 (0.49) HSD17B10CYP1A2CYP2D6CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed