SCHEMBL3400465

SCHEMBL3400465

Cc1nc(-c2ccccc2C(C)C)sc1C(=O)NCCCCN1CCCC1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SMYD2 Q9NRG4 8/20 0.47
GAA P10253 1/20 0.45
DRD3 P35462 3/20 0.42
DRD2 P14416 2/20 0.42
CHRM4 P08173 1/20 0.42
NPC1 O15118 1/20 0.42
HPGD P15428 1/20 0.42
HTR2C P28335 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
HTR1A P08908 1/20 0.41
HTR2A P28223 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3403455 0.93 PARP1 (0.46) SMYD2GAACHRM4NPC1HPGD
SCHEMBL3401847 0.92 HTR2C (0.45) SMYD2GAACHRM4NPC1HPGD
SCHEMBL3403787 0.87 SMYD2 (0.50) SMYD2GAADRD3DRD2CHRM4
SCHEMBL3403830 0.85 HTR3A (0.47) SMYD2GAADRD3DRD2L3MBTL1
SCHEMBL3405123 0.85 HTR3A (0.55) SMYD2DRD3DRD2HTR2CHTR1A
SCHEMBL3404056 0.85 PPARD (0.52) SMYD2GAADRD3DRD2CHRM4
SCHEMBL3402446 0.84 RAB9A (0.47) NPC1HPGDL3MBTL1
SCHEMBL3402982 0.83 SMYD2 (0.53) SMYD2GAACHRM4NPC1
SCHEMBL3396859 0.83 DRD2 (0.51) SMYD2GAADRD3DRD2HTR2C
SCHEMBL3404866 0.83 MCHR1 (0.46) SMYD2GAADRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed