SCHEMBL3400860

SCHEMBL3400860

Cc1nc(-c2ccccc2C(F)(F)F)sc1C(=O)NCCN1CCCCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 1/20 0.54
PPARA Q07869 1/20 0.54
CHRM4 P08173 3/20 0.49
HTR2C P28335 1/20 0.45
PARP1 P09874 1/20 0.45
POLB P06746 1/20 0.44
TSHR P16473 1/20 0.44
ACP1 P24666 1/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 1/20 0.44
NPY1R P25929 1/20 0.44
NPY2R P49146 1/20 0.44
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA4 P43681 1/20 0.43
NPC1 O15118 1/20 0.43
HPGD P15428 1/20 0.43
APP P05067 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3405687 0.99 PPARD (0.54) PPARDPPARACHRM4HTR2CPARP1
SCHEMBL3404913 0.93 PPARD (0.53) PPARDPPARACHRM4HTR2CACP1
SCHEMBL3404056 0.92 PPARD (0.52) PPARDPPARACHRM4ACP1SMYD2
SCHEMBL3401416 0.86 NPC1 (0.53) PPARDPPARACHRM4HTR2CPARP1
SCHEMBL3402762 0.85 NPC1 (0.53) PPARDPPARACHRM4HTR2CPARP1
SCHEMBL3401847 0.84 HTR2C (0.45) CHRM4HTR2CPARP1POLBKDM4E
SCHEMBL3403561 0.83 WNT1 (0.52) CHRM4HTR2CPARP1POLBTSHR
SCHEMBL3403455 0.83 PARP1 (0.46) CHRM4HTR2CPARP1POLBKDM4E
SCHEMBL3405526 0.83 PPARD (0.53) PPARDPPARACHRM4HTR2CNPC1
SCHEMBL3405595 0.82 PDE2A (0.47) PPARDPPARACHRM4HTR2CPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed