SCHEMBL3402010

SCHEMBL3402010

COc1ccc(Br)cc1C(=O)NC1COCCn2c1nc(-c1ccncn1)cc2=O

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 15/20 0.39
CYP2D6 P10635 6/20 0.39
CYP1A2 P05177 4/20 0.39
MTOR P42345 2/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3400870 0.92 GSK3B (0.42) GSK3BCYP2D6CYP1A2MTORCYP3A4
SCHEMBL3425658 0.91 KCNMA1 (0.40) GSK3BCYP2D6CYP1A2MTORALDH1A1
SCHEMBL3402173 0.90 GSK3B (0.45) GSK3BCYP2D6CYP1A2
SCHEMBL2064918 0.89 DRD2 (0.43) GSK3BCYP2D6CYP1A2ALDH1A1CYP3A4
SCHEMBL2065404 0.88 MEN1 (0.41) GSK3BCYP2D6CYP1A2ALDH1A1CYP3A4
SCHEMBL3402360 0.88 POLB (0.42) GSK3BCYP2D6CYP1A2ALDH1A1CYP2C19
SCHEMBL3661580 0.88 GSK3B (0.44) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL3402193 0.87 GSK3B (0.42) GSK3BCYP2D6CYP1A2MTORCYP3A4
SCHEMBL3399343 0.86 GSK3B (0.47) GSK3BCYP2D6CYP1A2MTOR
SCHEMBL3399573 0.86 GSK3B (0.44) GSK3BCYP2D6CYP1A2CYP3A4TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247599-A1 SUBSTITUTED ARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2010-11-10 EP claimed
WO-2009095788-A1 SUBSTITUTED ARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2009-08-06 WO claimed
EP-2247599-A1 SUBSTITUTED ARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2010-11-10 EP disclosed
WO-2009095788-A1 SUBSTITUTED ARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2009-08-06 WO disclosed