SCHEMBL3402360

SCHEMBL3402360

COc1ccc(S(N)(=O)=O)cc1C(=O)NC1COCCn2c1nc(-c1ccncn1)cc2=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.42
CA2 P00918 4/20 0.38
CYP1A2 P05177 3/20 0.38
CYP2D6 P10635 3/20 0.38
CA1 P00915 3/20 0.38
DRD2 P14416 2/20 0.38
DRD1 P21728 2/20 0.38
DRD4 P21917 2/20 0.38
DRD3 P35462 2/20 0.38
CA9 Q16790 2/20 0.38
CA12 O43570 2/20 0.38
CA7 P43166 2/20 0.38
MAPT P10636 2/20 0.38
CA3 P07451 1/20 0.38
ADRA2A P08913 1/20 0.38
PTGS1 P23219 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
BLM P54132 1/20 0.38
CA5B Q9Y2D0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2066169 0.89 POLB (0.49) POLBCA2CYP1A2CYP2D6CA1
SCHEMBL3400870 0.89 GSK3B (0.42) CYP1A2CYP2D6GSK3B
SCHEMBL3402010 0.88 GSK3B (0.39) CYP1A2CYP2D6CYP2C19KMT2AMEN1
SCHEMBL3425658 0.88 KCNMA1 (0.40) POLBCYP1A2CYP2D6MAPTKMT2A
SCHEMBL3402173 0.87 GSK3B (0.45) CYP1A2CYP2D6GSK3B
SCHEMBL3399684 0.85 CRBN (0.42) CYP1A2CYP2D6GSK3B
SCHEMBL3400823 0.85 HTR4 (0.42) CYP1A2CYP2D6DRD2DRD4DRD3
SCHEMBL3402193 0.84 GSK3B (0.42) CYP1A2CYP2D6LMNAGSK3B
SCHEMBL3399573 0.84 GSK3B (0.44) CYP1A2CYP2D6MAPTGSK3B
SCHEMBL3399343 0.84 GSK3B (0.47) CYP1A2CYP2D6GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247599-A1 SUBSTITUTED ARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2010-11-10 EP disclosed
WO-2009095788-A1 SUBSTITUTED ARYLAMIDE OXAZEPINOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2009-08-06 WO disclosed