SCHEMBL3401682

SCHEMBL3401682

Cc1cc(Cl)ccc1-c1cc2c(c(Nc3ccc(N4CCOCC4)cc3)n1)CNC=N2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ZAP70 P43403 2/20 0.44
CYP1B1 Q16678 2/20 0.43
CYP1A2 P05177 1/20 0.43
ALOX5 P09917 1/20 0.41
MAPT P10636 6/20 0.41
MAPK1 P28482 3/20 0.41
TP53 P04637 1/20 0.41
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40
GAA P10253 3/20 0.40
LMNA P02545 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
TACR2 P21452 2/20 0.40
RECQL P46063 1/20 0.40
PLK4 O00444 2/20 0.40
ALDH1A1 P00352 1/20 0.39
PTK2B Q14289 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3402080 0.88 ZAP70 (0.48) ZAP70CYP1B1CYP1A2ALOX5MAPT
SCHEMBL3397387 0.84 ZAP70 (0.48) ZAP70CYP1B1CYP1A2ALOX5MAPT
SCHEMBL3405873 0.81 ZAP70 (0.46) ZAP70CYP1B1CYP1A2ALOX5MAPT
SCHEMBL3397301 0.79 MAPT (0.50) ZAP70CYP1A2MAPTMAPK1TP53
SCHEMBL3428156 0.76 ZAP70 (0.45) ZAP70ALOX5MAPTMAPK1GAA
SCHEMBL3428992 0.76 AURKA (0.49) ZAP70MAPTMAPK1TP53NPSR1
SCHEMBL3406123 0.75 IGF1R (0.48) ZAP70MAPTMAPK1TP53GAA
SCHEMBL1059221 0.74 SYK (0.57) ZAP70MAPTGAALMNAMEN1
SCHEMBL3394570 0.69 ZAP70 (0.55) ZAP70CYP1B1MAPTMAPK1GAA
SCHEMBL3359711 0.66 MAPT (0.42) ZAP70CYP1B1CYP1A2ALOX5MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250169-A1 PYRIDO [4, 3-D]PYRIMIDINONE DERIVATIVES AS KINASE INHIBITORS IRM LLC (BM) 2010-11-17 EP claimed
WO-2009099801-A1 PYRIDO [4, 3-D] PYRIMIDINONE DERIVATIVES AS KINASE INHIBITORS IRM LLC (BM) 2009-08-13 WO claimed