SCHEMBL3402500

SCHEMBL3402500

CNCC(=O)N(C)CC(C)C

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PYGL P06737 1/20 0.39
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
MEN1 O00255 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
CACNA1H O95180 1/20 0.30
KDM4C Q9H3R0 2/20 0.30
KDM4A O75164 1/20 0.30
PHF8 Q9UPP1 1/20 0.30
KDM2A Q9Y2K7 1/20 0.30
NAMPT P43490 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22951198 0.83 PYGL (0.39) PYGLCA12CA1CA2CA9
SCHEMBL22305724 0.81 PYGL (0.38) PYGLCA12CA1CA2CA9
SCHEMBL3402497 0.78 ADH1B (0.40) PYGLCA12CA1CA2CA9
SCHEMBL8623620 0.77 CA1 (0.41) PYGLCA12CA1CA2CA9
SCHEMBL12227388 0.75 CA12 (0.42) CA12CA1CA2CA9
SCHEMBL17689169 0.75 PYGL (0.40) PYGLCA12CA1CA2CA9
SCHEMBL14930120 0.75
SCHEMBL12734485 0.75 ALDH1A1 (0.42) PYGLCA12CA1CA2CA9
SCHEMBL3402498 0.74 CA12 (0.35) PYGLCA12CA1CA2CA9
SCHEMBL12253911 0.74 CA12 (0.35) PYGLCA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8394789-B2 (Dihydro)pyrrolo[2,1-α]isoquinolines MSD OSS B.V. (NL) 2013-03-12 US disclosed
EP-2252611-A1 (DIHYDRO)PYRROLO[2,1-A]ISOQUINOLINES N.V. Organon (NL) 2010-11-24 EP disclosed
WO-2009098283-A1 (DIHYDRO)PYRROLO[2,1-A]ISOQUINOLINES N.V. ORGANON (NL) 2009-08-13 WO disclosed