SCHEMBL3402497

SCHEMBL3402497

CC(C)CN(C)C(=O)CNC=O

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADH1B P00325 1/20 0.40
ADH1C P00326 1/20 0.40
ADH1A P07327 1/20 0.40
PYGL P06737 1/20 0.36
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22951198 0.78 PYGL (0.39) PYGLCA12CA1CA2CA9
SCHEMBL3402500 0.78 PYGL (0.39) PYGLCA12CA1CA2CA9
SCHEMBL22305724 0.76 PYGL (0.38) PYGLCA12CA1CA2CA9
SCHEMBL22114486 0.76 ADH1B (0.38) ADH1BADH1CADH1ALMNA
SCHEMBL3075746 0.74
SCHEMBL19751307 0.74 MVD (0.38) LMNA
SCHEMBL24738913 0.73 LMNA (0.30) LMNA
SCHEMBL8623620 0.72 CA1 (0.41) PYGLCA12CA1CA2CA9
SCHEMBL17689169 0.70 PYGL (0.40) PYGLCA12CA1CA2CA9
SCHEMBL12734485 0.70 ALDH1A1 (0.42) PYGLCA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8394789-B2 (Dihydro)pyrrolo[2,1-α]isoquinolines MSD OSS B.V. (NL) 2013-03-12 US disclosed
EP-2252611-A1 (DIHYDRO)PYRROLO[2,1-A]ISOQUINOLINES N.V. Organon (NL) 2010-11-24 EP disclosed
WO-2009098283-A1 (DIHYDRO)PYRROLO[2,1-A]ISOQUINOLINES N.V. ORGANON (NL) 2009-08-13 WO disclosed