SCHEMBL3403501

SCHEMBL3403501

CCn1cc(C(=O)OC2CC2)c(=O)c2cc(F)c(F)c(OCC[C@H]3C[C@@H](O[Si](C)(C)C(C)(C)C)CN3C(=O)OCc3ccccc3)c21

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 1/20 0.35
TSHR P16473 3/20 0.34
MAPK1 P28482 1/20 0.34
TOP1 P11387 5/20 0.34
ALDH1A1 P00352 4/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KDM4E B2RXH2 4/20 0.31
HPGD P15428 3/20 0.31
HSD17B10 Q99714 3/20 0.31
PDK1 Q15118 1/20 0.31
PDK2 Q15119 1/20 0.31
PDK3 Q15120 1/20 0.31
PDK4 Q16654 1/20 0.31
PMP22 Q01453 1/20 0.31
TDP1 Q9NUW8 1/20 0.30
LMNA P02545 1/20 0.30
ABCB1 P08183 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL143025 0.88 ADRB2 (0.40) STAT3ALDH1A1KDM4EHPGDTDP1
SCHEMBL143026 0.81 AGTR2 (0.30)
SCHEMBL115725 0.75 ADRB2 (0.43) STAT3ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL12825630 0.71 ADRB2 (0.40) STAT3ALDH1A1KDM4EHPGDPDK1
SCHEMBL115984 0.71 PDK1 (0.43) PDK1PDK2PDK3PDK4ABCB1
SCHEMBL12825261 0.70 ADRB2 (0.43) STAT3ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL3820416 0.70 TOP1 (0.44) STAT3TOP1ALDH1A1KDM4EHPGD
SCHEMBL1461785 0.69 KDM4E (0.40) STAT3TSHRTOP1ALDH1A1KDM4E
SCHEMBL583954 0.69 STAT3 (0.43) STAT3TSHRMAPK1TOP1ALDH1A1
SCHEMBL10390664 0.69 ABCB1 (0.41) ALDH1A1KDM4EPDK1PDK2PDK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250171-A2 ANTIBACTERIAL FLUOROQUINOLONE ANALOGS Achaogen, Inc. (US) 2010-11-17 EP disclosed
WO-2009137130-A2 ANTIBACTERIAL FLUOROQUINOLONE ANALOGS ACHAOGEN, INC. (US) 2009-11-12 WO disclosed