SCHEMBL3403592

SCHEMBL3403592

CCOc1cccc(-c2nc(C)c(C(=O)N(CC)CCN(C)CC)s2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
HPGD P15428 3/20 0.42
KDM4E B2RXH2 2/20 0.42
HSD17B10 Q99714 2/20 0.42
TRPM8 Q7Z2W7 3/20 0.42
NOTUM Q6P988 1/20 0.42
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 4/20 0.40
RAB9A P51151 2/20 0.40
NPC1 O15118 2/20 0.40
MEN1 O00255 1/20 0.40
TP53 P04637 1/20 0.40
PPARD Q03181 2/20 0.39
PPARA Q07869 2/20 0.39
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
USP2 O75604 1/20 0.39
CDC7 O00311 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3404830 0.88 ALDH1A1 (0.44) ALDH1A1HPGDTRPM8KMT2ASMN1; SMN2
SCHEMBL3403251 0.87 SMN1; SMN2 (0.46) ALDH1A1HPGDTRPM8KMT2ASMN1; SMN2
SCHEMBL3401041 0.85 TRPM8 (0.53) ALDH1A1TRPM8KMT2ASMN1; SMN2RAB9A
SCHEMBL3404718 0.85 KMT2A (0.60) ALDH1A1HPGDKDM4ETRPM8KMT2A
SCHEMBL3402129 0.84 HTR2C (0.43) ALDH1A1HPGDKDM4ETRPM8KMT2A
SCHEMBL3397100 0.83 HTR2C (0.46) ALDH1A1HPGDKDM4EHSD17B10TRPM8
SCHEMBL3399358 0.83 ALDH1A1 (0.43) ALDH1A1HPGDTRPM8KMT2ASMN1; SMN2
SCHEMBL3402204 0.83 KMT2A (0.42) ALDH1A1HPGDTRPM8KMT2ASMN1; SMN2
SCHEMBL3403795 0.82 NPC1 (0.47) ALDH1A1HPGDKDM4ETRPM8KMT2A
SCHEMBL3405333 0.81 RAB9A (0.40) ALDH1A1HPGDKDM4ETRPM8KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed