SCHEMBL3406028

SCHEMBL3406028

CCCOc1ccc(-c2nc(C)c(C(=O)NCCN3CCCC3)s2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
NPC1 O15118 1/20 0.47
HPGD P15428 1/20 0.47
POLB P06746 1/20 0.47
CHRM4 P08173 3/20 0.47
HRH3 Q9Y5N1 1/20 0.46
SCN9A Q15858 1/20 0.46
MAPT P10636 4/20 0.45
AGER Q15109 3/20 0.45
ALDH1A1 P00352 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
HSD17B10 Q99714 1/20 0.45
KMT2A Q03164 1/20 0.45
THRB P10828 1/20 0.45
TSHR P16473 1/20 0.45
PPARA Q07869 2/20 0.45
TARBP2 Q15633 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3401121 0.94 AGER (0.47) NPC1HPGDCHRM4HRH3MAPT
SCHEMBL3405206 0.92 GLA (0.60) GLAL3MBTL1NPC1HPGDPOLB
SCHEMBL3398904 0.89 POLB (0.60) NPC1HPGDPOLBCHRM4SCN9A
SCHEMBL3398969 0.86 HPGD (0.55) NPC1HPGDPOLBCHRM4SCN9A
SCHEMBL3398806 0.85 CHRM4 (0.54) NPC1HPGDPOLBCHRM4SCN9A
SCHEMBL3401424 0.85 PPARA (0.61) NPC1POLBCHRM4SCN9AALDH1A1
SCHEMBL13310379 0.84 ACKR3 (0.50) NPC1HPGDCHRM4HRH3MAPT
SCHEMBL3405464 0.84 PPARA (0.60) NPC1POLBCHRM4SCN9AALDH1A1
SCHEMBL3398394 0.83 KDM4E (0.54) POLBCHRM4SCN9AMAPTALDH1A1
SCHEMBL3404512 0.83 HRH3 (0.62) NPC1CHRM4HRH3CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed