SCHEMBL3404331

SCHEMBL3404331

COc1cc(Nc2cc(C(F)(F)F)cc(Nc3ccc(C(F)(F)F)cc3)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.41
ABCC1 P33527 3/20 0.41
ABCG2 Q9UNQ0 3/20 0.41
DHODH Q02127 1/20 0.41
GAK O14976 1/20 0.41
GALR2 O43603 1/20 0.40
PSEN1 P49768 3/20 0.39
PSEN2 P49810 3/20 0.39
APH1B Q8WW43 3/20 0.39
NCSTN Q92542 3/20 0.39
APH1A Q96BI3 3/20 0.39
PSENEN Q9NZ42 3/20 0.39
AGPAT2 O15120 1/20 0.39
DYRK1A Q13627 1/20 0.37
PLK1 P53350 1/20 0.36
TP53 P04637 1/20 0.36
BRAF P15056 3/20 0.35
TNIK Q9UKE5 1/20 0.35
RAF1 P04049 1/20 0.35
JAK2 O60674 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3404327 0.93 DHODH (0.43) ABCB1ABCC1ABCG2DHODHGAK
SCHEMBL3410953 0.93 ABCB1 (0.44) ABCB1ABCC1ABCG2DHODHGAK
SCHEMBL3404287 0.91 GALR2 (0.41) ABCB1ABCC1ABCG2GAKGALR2
SCHEMBL3409746 0.91 TP53 (0.47) ABCB1ABCC1ABCG2PSEN1PSEN2
SCHEMBL3412202 0.91 MAPT (0.42) ABCB1ABCC1ABCG2GAKGALR2
SCHEMBL3410067 0.87 IGF1R (0.47) ABCB1ABCC1ABCG2GAKGALR2
SCHEMBL3413181 0.86 TP53 (0.48) ABCB1ABCC1ABCG2PSEN1PSEN2
SCHEMBL3406352 0.81 BRAF (0.46) ABCB1ABCC1ABCG2PSEN1PSEN2
SCHEMBL3407803 0.81 IGF1R (0.43) ABCB1ABCC1ABCG2GALR2BRAF
SCHEMBL3409749 0.81 IMPDH2 (0.42) ABCB1ABCC1ABCG2GAKPSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed