SCHEMBL3406372

SCHEMBL3406372

O=C(NC1CCCCn2c1nc(-c1ccncc1)cc2=O)c1[c]cccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CGAS Q8N884 1/20 0.37
CYP2C9 P11712 2/20 0.36
GSK3B P49841 10/20 0.36
CDC7 O00311 2/20 0.35
MAP4K4 O95819 2/20 0.35
PIM1 P11309 2/20 0.35
PRKACA P17612 2/20 0.35
CDK2 P24941 2/20 0.35
HIPK2 Q9H2X6 2/20 0.35
CLK4 Q9HAZ1 2/20 0.35
IRAK4 Q9NWZ3 2/20 0.35
ROCK2 O75116 3/20 0.35
ROCK1 Q13464 3/20 0.35
DYRK3 O43781 1/20 0.35
CDK1 P06493 1/20 0.35
CSF1R P07333 1/20 0.35
MARK3 P27448 1/20 0.35
MAPK1 P28482 1/20 0.35
CSNK1A1 P48729 1/20 0.35
CSNK1D P48730 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3400978 0.89 GSK3B (0.39) GSK3BCYP1A2CYP2D6
SCHEMBL3401659 0.86 GSK3B (0.39) GSK3BCYP1A2CYP2D6
SCHEMBL4390474 0.81 ALDH1A1 (0.46) GSK3BKDM4EHTT
SCHEMBL2065962 0.80 KMT2A (0.46) CGASGSK3BKDM4E
SCHEMBL2065321 0.79 KDM4E (0.43) KDM4E
SCHEMBL2066118 0.79 ALDH1A1 (0.43) CGASGSK3BCYP1A2
SCHEMBL2065004 0.79 PRKACA (0.47) GSK3BCDC7MAP4K4PIM1PRKACA
SCHEMBL4391863 0.79 MAPT (0.40) CGASCYP2C9GSK3BCDC7MAP4K4
SCHEMBL4391283 0.79 CYP2C9 (0.39) CGASCYP2C9GSK3BCDC7MAP4K4
SCHEMBL4386108 0.79 RAB9A (0.41) GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957492-B1 SUBSTITUTED BICYCLIC PYRIMIDONE DERIVATIVES SANOFI AVENTIS (FR) 2010-11-10 EP claimed