SCHEMBL3406645

SCHEMBL3406645

COc1cc(Nc2nc(-c3cccs3)cc(C(C)(C)O)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.37
TP53 P04637 4/20 0.37
MAPT P10636 9/20 0.36
SMPD3 Q9NY59 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
ABCB1 P08183 1/20 0.35
ABCC1 P33527 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35
TLR8 Q9NR97 1/20 0.35
MEN1 O00255 5/20 0.35
KMT2A Q03164 5/20 0.35
KDM4E B2RXH2 4/20 0.35
RAB9A P51151 4/20 0.35
NPC1 O15118 3/20 0.35
NFKB1 P19838 3/20 0.35
NFKB2 Q00653 3/20 0.35
RELA Q04206 3/20 0.35
GAA P10253 2/20 0.35
SHMT2 P34897 1/20 0.35
ALDH1A1 P00352 5/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3408862 0.84 NPC1 (0.43) ABCG2MEN1KMT2AKDM4ERAB9A
SCHEMBL3406823 0.83 NPC1 (0.39) SMN1; SMN2MAPTRAB9ANPC1GAA
SCHEMBL3406534 0.83 SYK (0.39) ABCB1ABCG2IMPDH2
SCHEMBL3410560 0.83 NPC1 (0.37) MAPTABCG2RAB9ANPC1GAA
SCHEMBL3412354 0.83 PTGS2 (0.39) SMN1; SMN2TP53MAPTKDM4EALDH1A1
SCHEMBL3409683 0.83 KMT2A (0.40) SMN1; SMN2TP53MAPTTDP1MEN1
SCHEMBL3409722 0.82 PIK3CA (0.41) SMN1; SMN2TP53MAPTRAB9ANPC1
SCHEMBL3412384 0.82 AGPAT2 (0.41) MAPTRAB9ANPC1GAA
SCHEMBL3405215 0.82 KCNH2 (0.37) RAB9ANPC1IMPDH2
SCHEMBL3410112 0.81 PSEN1 (0.36) MAPTABCG2MEN1KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed