SCHEMBL3407602

SCHEMBL3407602

CN(C)C1(c2ccccc2)CCC(c2ccccc2)(N(C)C(=O)Oc2cccnc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 18/20 0.55
OPRL1 P41146 17/20 0.55
OPRK1 P41145 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4344674 0.79 OPRM1 (0.62) OPRM1OPRL1OPRK1
SCHEMBL23778868 0.74 OPRM1 (0.51) OPRM1OPRL1OPRK1
SCHEMBL10635171 0.74 RAB9A (0.57)
SCHEMBL31524305 0.74 RAB9A (0.57)
SCHEMBL23778489 0.73 OPRM1 (0.41) OPRM1OPRL1
SCHEMBL5648895 0.73 LIPE (0.56)
SCHEMBL12521051 0.72 OPRM1 (0.65) OPRM1OPRL1OPRK1
SCHEMBL3410403 0.72 OPRM1 (1.00) OPRM1OPRL1OPRK1
SCHEMBL20904051 0.69 OPRM1 (0.59) OPRM1OPRL1OPRK1
SCHEMBL28140609 0.69 KMT2A (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2502907-A1 Substituted 4-aminocyclohexane derivatives Grünenthal GmbH (DE) 2012-09-26 EP claimed
EP-2260021-A1 SUBSTITUTED 4-AMINOCYCLOHEXANE DERIVATIVES Grünenthal GmbH (DE) 2010-12-15 EP claimed
WO-2009118168-A1 SUBSTITUTED 4-AMINOCYCLOHEXANE DERIVATIVES Grünenthal GmbH (DE) 2009-10-01 WO claimed
EP-2502907-B1 Substituted 4-aminocyclohexane derivatives GRUENENTHAL GMBH (DE) 2018-08-29 EP disclosed
EP-2518052-B1 Substituted 4-aminocyclohexane derivatives GRUENENTHAL GMBH (DE) 2017-12-20 EP disclosed
EP-2260021-B1 SUBSTITUTED 4-AMINOCYCLOHEXANE DERIVATIVES GRUENENTHAL GMBH (DE) 2014-04-23 EP disclosed
EP-2518052-A1 Substituted 4-aminocyclohexane derivatives Grünenthal GmbH (DE) 2012-10-31 EP disclosed
EP-2502907-A1 Substituted 4-aminocyclohexane derivatives Grünenthal GmbH (DE) 2012-09-26 EP disclosed