SCHEMBL3410440

SCHEMBL3410440

COc1cc(Nc2nc(Cl)cc(CC(C)c3ccc(Cl)cc3)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
AGPAT2 O15120 4/20 0.35
PLK1 P53350 1/20 0.33
KCNH2 Q12809 1/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
MAPT P10636 3/20 0.32
GAA P10253 1/20 0.32
IMPDH2 P12268 2/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
KMT2A Q03164 1/20 0.32
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
KDR P35968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3413396 0.89 PIK3CA (0.39) NPC1RAB9APLK1PSEN1PSEN2
SCHEMBL3410239 0.83 KDR (0.38) NPC1RAB9APLK1PSEN1PSEN2
SCHEMBL3407955 0.81 NPC1 (0.51) NPC1RAB9AKCNH2MAPTGAA
SCHEMBL3406232 0.81 NPC1 (0.41) NPC1RAB9AKCNH2PSEN1PSEN2
SCHEMBL3413207 0.78 PSEN1 (0.52) NPC1RAB9AAGPAT2KCNH2PSEN1
SCHEMBL3408338 0.77 NPC1 (0.40) NPC1RAB9APLK1KCNH2PSEN1
SCHEMBL3408813 0.77 SYK (0.35) PLK1KDRSTK17AP2RX3
SCHEMBL3412730 0.76 PIK3CA (0.40) NPC1RAB9AAGPAT2KCNH2PSEN1
SCHEMBL3410260 0.76 NPC1 (0.53) NPC1RAB9AKCNH2MAPTGAA
SCHEMBL3412452 0.76 EGFR (0.40) SMN1; SMN2KDRSTK17A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed