SCHEMBL3407955

SCHEMBL3407955

COc1cc(Nc2nc(C)cc(Cl)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
KCNH2 Q12809 1/20 0.43
DOT1L Q8TEK3 1/20 0.41
MAPT P10636 3/20 0.41
GAA P10253 1/20 0.41
BRD4 O60885 1/20 0.40
IMPDH2 P12268 3/20 0.39
EHMT2 Q96KQ7 4/20 0.38
EHMT1 Q9H9B1 4/20 0.38
TERT O14746 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
LMNA P02545 1/20 0.37
EPHB4 P54760 1/20 0.37
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3410260 0.92 NPC1 (0.53) NPC1RAB9AKCNH2DOT1LMAPT
SCHEMBL3406068 0.87 NPC1 (0.46) NPC1RAB9AKCNH2DOT1LMAPT
SCHEMBL3408803 0.85 MEN1 (0.46) NPC1RAB9AKCNH2DOT1LIMPDH2
SCHEMBL3410316 0.85 IMPDH2 (0.44) NPC1RAB9AKCNH2DOT1LMAPT
SCHEMBL3411066 0.84 NPC1 (0.47) NPC1RAB9AKCNH2DOT1LMAPT
SCHEMBL3410885 0.84 NPC1 (0.44) NPC1RAB9AKCNH2DOT1LMAPT
SCHEMBL3408862 0.84 NPC1 (0.43) NPC1RAB9AKCNH2DOT1LBRD4
SCHEMBL3410702 0.83 USP2 (0.45) NPC1RAB9AKCNH2DOT1LMAPT
SCHEMBL3409949 0.83 IMPDH2 (0.51) NPC1RAB9AKCNH2DOT1LIMPDH2
SCHEMBL3411085 0.83 NPC1 (0.42) NPC1RAB9AKCNH2DOT1LMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed