SCHEMBL3410885

SCHEMBL3410885

COc1cc(Nc2nc(C)cc(Oc3ccc(Cl)cc3)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
KCNH2 Q12809 1/20 0.40
TSHR P16473 1/20 0.39
AGPAT2 O15120 2/20 0.38
SCN9A Q15858 2/20 0.38
SCN5A Q14524 1/20 0.38
MAPK1 P28482 1/20 0.36
SLC2A1 P11166 1/20 0.36
DOT1L Q8TEK3 1/20 0.36
BRD4 O60885 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ATM Q13315 1/20 0.36
MAPT P10636 2/20 0.35
GAA P10253 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3406468 0.90 KCNH2 (0.42) NPC1RAB9AKCNH2DOT1LCYP1A2
SCHEMBL3410450 0.89 NPC1 (0.38) NPC1RAB9AKCNH2DOT1LCYP1A2
SCHEMBL3412873 0.89 KCNH2 (0.45) NPC1RAB9AKCNH2SCN9AMAPK1
SCHEMBL3413137 0.88 CHRNA7 (0.40) NPC1RAB9AKCNH2SCN9ASCN5A
SCHEMBL3413260 0.88 GAK (0.39) NPC1RAB9AKCNH2SCN9AMAPK1
SCHEMBL3406068 0.87 NPC1 (0.46) NPC1RAB9AKCNH2TSHRDOT1L
SCHEMBL3410260 0.84 NPC1 (0.53) NPC1RAB9AKCNH2MAPK1DOT1L
SCHEMBL3410439 0.84 SCN9A (0.41) AGPAT2SCN9A
SCHEMBL3407955 0.84 NPC1 (0.51) NPC1RAB9AKCNH2DOT1LBRD4
SCHEMBL3410139 0.83 EGFR (0.46) NPC1RAB9AKCNH2SCN9ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed