SCHEMBL3406068

SCHEMBL3406068

COc1cc(C)nc(Nc2ccc(-c3nc(C)c[nH]3)c(OC)c2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
KCNH2 Q12809 1/20 0.44
IMPDH2 P12268 4/20 0.43
DOT1L Q8TEK3 1/20 0.42
HTT P42858 1/20 0.39
EHMT2 Q96KQ7 4/20 0.39
EHMT1 Q9H9B1 4/20 0.39
TERT O14746 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
BRD4 O60885 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3410316 0.95 IMPDH2 (0.44) NPC1RAB9AKCNH2IMPDH2DOT1L
SCHEMBL3410260 0.93 NPC1 (0.53) NPC1RAB9AKCNH2IMPDH2DOT1L
SCHEMBL3410702 0.90 USP2 (0.45) NPC1RAB9AKCNH2IMPDH2DOT1L
SCHEMBL3411085 0.90 NPC1 (0.42) NPC1RAB9AKCNH2IMPDH2DOT1L
SCHEMBL3406681 0.88 NPC1 (0.41) NPC1RAB9AKCNH2IMPDH2DOT1L
SCHEMBL3407955 0.87 NPC1 (0.51) NPC1RAB9AKCNH2IMPDH2DOT1L
SCHEMBL3408568 0.87 NPC1 (0.39) NPC1RAB9AKCNH2IMPDH2DOT1L
SCHEMBL3410885 0.87 NPC1 (0.44) NPC1RAB9AKCNH2IMPDH2DOT1L
SCHEMBL3406468 0.87 KCNH2 (0.42) NPC1RAB9AKCNH2IMPDH2DOT1L
SCHEMBL3412405 0.86 NPC1 (0.39) NPC1RAB9AKCNH2IMPDH2DOT1L

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed