SCHEMBL3412873

SCHEMBL3412873

COc1cc(Nc2nc(C)cc(Oc3ccc(F)c(F)c3)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.45
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
APP P05067 1/20 0.36
DOT1L Q8TEK3 1/20 0.35
METAP2 P50579 1/20 0.34
GALR2 O43603 3/20 0.34
IMPDH2 P12268 3/20 0.34
GALR1 P47211 1/20 0.34
EHMT2 Q96KQ7 3/20 0.33
EHMT1 Q9H9B1 3/20 0.33
PARP1 P09874 1/20 0.33
KDR P35968 1/20 0.33
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33
TUBB4B P68371 1/20 0.33
TUBB3 Q13509 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3406468 0.91 KCNH2 (0.42) KCNH2NPC1RAB9ADOT1LIMPDH2
SCHEMBL3410885 0.89 NPC1 (0.44) KCNH2NPC1RAB9AAPPDOT1L
SCHEMBL3413260 0.86 GAK (0.39) KCNH2NPC1RAB9AAPPDOT1L
SCHEMBL3413137 0.86 CHRNA7 (0.40) KCNH2NPC1RAB9ADOT1LGALR2
SCHEMBL3410450 0.85 NPC1 (0.38) KCNH2NPC1RAB9ADOT1LIMPDH2
SCHEMBL3406068 0.85 NPC1 (0.46) KCNH2NPC1RAB9ADOT1LIMPDH2
SCHEMBL3411030 0.84 MAPT (0.41) KCNH2NPC1RAB9AAPPLMNA
SCHEMBL3410260 0.83 NPC1 (0.53) KCNH2NPC1RAB9ADOT1LIMPDH2
SCHEMBL3413250 0.82 SLC2A1 (0.42) NPC1RAB9ALMNAHTTSLC2A1
SCHEMBL3410316 0.81 IMPDH2 (0.44) KCNH2NPC1RAB9ADOT1LIMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed