SCHEMBL3415853

SCHEMBL3415853

C=C(N)NS(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.57
CA2 P00918 3/20 0.57
MMP2 P08253 2/20 0.57
MMP1 P03956 1/20 0.57
MMP9 P14780 1/20 0.57
MMP8 P22894 1/20 0.57
MMP13 P45452 1/20 0.57
F2 P00734 1/20 0.56
PRSS1 P07477 1/20 0.56
PRSS2 P07478 1/20 0.56
PRSS3 P35030 1/20 0.56
GAA P10253 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
ALDH1A1 P00352 2/20 0.51
CA9 Q16790 3/20 0.51
CA12 O43570 2/20 0.51
CA14 Q9ULX7 2/20 0.51
NPSR1 Q6W5P4 1/20 0.51
CA4 P22748 1/20 0.51
CA6 P23280 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18296817 0.82 TSHR (0.61) CA1CA2MMP2MMP1MMP9
SCHEMBL170426 0.82 CA1 (0.59) CA1CA2MMP2MMP1MMP9
SCHEMBL12968291 0.82 MMP2 (0.59) CA1CA2MMP2MMP1MMP9
SCHEMBL8038636 0.81 CA1 (0.57) CA1CA2MMP2MMP1MMP9
SCHEMBL7363066 0.81 ALDH1A1 (0.60) CA1CA2MMP2MMP1MMP9
SCHEMBL29135554 0.79 LMNA (0.58) CA1CA2MMP2MMP1MMP9
SCHEMBL21561788 0.79 NPSR1 (0.58) CA1CA2MMP2MMP1MMP9
SCHEMBL5177115 0.79 NPSR1 (0.50) CA1CA2MMP2MMP1MMP9
SCHEMBL195196 0.78 LMNA (0.56) CA1CA2MMP2MMP1MMP9
SCHEMBL19011399 0.78 MMP2 (0.53) CA1CA2MMP2MMP1MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2152715-B1 IMPROVED PROCESS FOR THE PREPARATION OF 6-ALPHA-HYDROXY-N-ALKYLATED OPIATES MALLINCKRODT INC (US) 2010-12-29 EP claimed