SCHEMBL3417508

SCHEMBL3417508

c1cnc2nc3conc3cc2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
POLB P06746 1/20 0.36
KDM4E B2RXH2 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
LMNA P02545 2/20 0.35
CASP6 P55212 1/20 0.35
HTT P42858 3/20 0.34
CASP1 P29466 2/20 0.34
TP53 P04637 2/20 0.34
HSP90AA1 P07900 2/20 0.34
MAPT P10636 2/20 0.34
TSHR P16473 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
CASP7 P55210 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
NR4A2 P43354 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20272946 0.77 ALDH1A1 (0.44) ALDH1A1NPC1RAB9APOLBKDM4E
SCHEMBL997757 0.75 ALDH1A1 (0.54) ALDH1A1NPC1RAB9APOLBKDM4E
SCHEMBL9824798 0.74 LMNA (0.40) NPC1RAB9APOLBKDM4ELMNA
SCHEMBL13156531 0.73 ALDH1A1 (0.46) ALDH1A1NPC1RAB9APOLBKDM4E
SCHEMBL3664517 0.72
SCHEMBL8170243 0.72 ALDH1A1 (0.54) ALDH1A1NPC1RAB9APOLBKDM4E
SCHEMBL3386562 0.71 ALDH1A1 (0.41) ALDH1A1NPC1RAB9APOLBKDM4E
SCHEMBL29384237 0.71 ALDH1A1 (0.48) ALDH1A1NPC1RAB9APOLBKDM4E
SCHEMBL832575 0.71 ALDH1A1 (0.48) ALDH1A1NPC1RAB9APOLBKDM4E
SCHEMBL28910441 0.71 ALDH1A1 (0.48) ALDH1A1NPC1RAB9APOLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1848723-B1 NEW ISOTHIAZOLOQUINOLONES AND RELATED COMPOUNDS AS ANTI-INFECTIVE AGENTS ACHILLION PHARMACEUTICALS INC (US) 2010-12-15 EP disclosed
EP-0227088-B1 ISOXAZOLO-NAPHTHYRIDINE, ISOXAZOLO QUINOLINE, ISOTHIAZOLONAPHTHYRIDINE, AND ISOTHIAZOLOQUINOLINE DERIVATIVES ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
EP-0227088-B1 ISOXAZOLO-NAPHTHYRIDINE, ISOXAZOLO QUINOLINE, ISOTHIAZOLONAPHTHYRIDINE, AND ISOTHIAZOLOQUINOLINE DERIVATIVES ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
US-4880814-A 7-cycloalkyl naphthyridines ABBOTT LABORATORIES (US) 1989-11-14 US disclosed
US-4767762-A Tricyclic quinoline and naphthyride antibacterials ABBOTT LABORATORIES (US) 1988-08-30 US disclosed
US-4767762-A Tricyclic quinoline and naphthyride antibacterials ABBOTT LABORATORIES (US) 1988-08-30 US disclosed
EP-0227088-A1 Isoxazolo-naphthyridine, isoxazolo quinoline, isothiazolonaphthyridine, and isothiazoloquinoline derivatives ABBOTT LABORATORIES (US) 1987-07-01 EP disclosed
EP-0227088-A1 Isoxazolo-naphthyridine, isoxazolo quinoline, isothiazolonaphthyridine, and isothiazoloquinoline derivatives ABBOTT LABORATORIES (US) 1987-07-01 EP disclosed