SCHEMBL3418103

SCHEMBL3418103

N#Cc1cc(F)ccc1C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.48
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
NOTUM Q6P988 1/20 0.41
POLB P06746 1/20 0.41
FFAR1 O14842 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
P4HB P07237 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1110956 0.85 KEAP1 (0.53) KEAP1CES2CES1NOTUMFFAR1
SCHEMBL17099949 0.83 CES2 (0.42) KEAP1CES2CES1POLBP4HB
SCHEMBL16051600 0.83 CYP1A2 (0.49) CES2CES1POLBP4HB
SCHEMBL16082919 0.79 PTPN1 (0.46) CES2CES1POLBFFAR1FFAR4
SCHEMBL30195093 0.79 PTPN1 (0.46) CES2CES1POLBFFAR1FFAR4
SCHEMBL162217 0.79 HPGD (0.53) POLBFFAR4
SCHEMBL4849617 0.78 XDH (0.50) NOTUMFFAR1
SCHEMBL19695306 0.78 ALDH1A1 (0.49) POLB
SCHEMBL30646082 0.78 CA9 (0.55) CES2POLB
SCHEMBL2832919 0.78 KEAP1 (0.46) KEAP1CES2CES1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2146753-A2 18F FLUORO-BENZOYL LABELLED BIOLOGICAL ACTIVE COMPOUNDS AS DIAGNOSTIC IMAGING AGENTS AS WELL AS BENZOTRIAZOL-1-YLOXY-BENZOYL , 2,5-DIOXO-PYRROLIDIN-1-YLOXY)BENZOYL AND TRIMETHYLAMMONIO-BENZOYL PRECURSERS THEREOF Bayer Schering Pharma Aktiengesellschaft (DE) 2010-01-27 EP disclosed
WO-2008104203-A2 18F FLUORO-BENZOYL LABELLED BIOLOGICAL ACTIVE COUMPOUNDS AS DIAGNOSITIC IMAGING AGENTS AS WELL AS BENZOTRIAZOL-1-YLOXY-BENZOYL, 2,5-DIOXO-PYRROLIDIN-1-YLOXY) BENZOYL AND TRIMETHYLAMMONIO-BENZOYL PRECURSERS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-09-04 WO disclosed