SCHEMBL3422378

SCHEMBL3422378

Cc1cccc(-n2cc(Cl)cn2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 6/20 0.48
GRIN1 Q05586 6/20 0.48
GRIN2B Q13224 6/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
PAX8 Q06710 1/20 0.48
GRM4 Q14833 1/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
ALPG P10696 1/20 0.41
CYP2C9 P11712 1/20 0.41
PKM P14618 1/20 0.41
ALOX12 P18054 1/20 0.41
NTSR1 P30989 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5110176 0.84 L3MBTL1 (0.46) RXRAGRIN1GRIN2BNPC1RAB9A
SCHEMBL13106298 0.82 RXRA (0.43) RXRAGRIN1GRIN2BRAB9AGRM4
SCHEMBL16789159 0.80 GRM4 (0.49) NPC1RAB9AGRM4KMT2AMEN1
SCHEMBL27822297 0.79 FAAH (0.40) NPC1RAB9AGRM4KMT2AMEN1
SCHEMBL9134471 0.79 NOTUM (0.47) RXRANPC1RAB9APAX8KMT2A
SCHEMBL23403693 0.79 GAA (0.62) RXRAGRIN1GRIN2BNPC1RAB9A
SCHEMBL22632940 0.79 KMT2A (0.47) RXRAGRIN1GRIN2BNPC1RAB9A
SCHEMBL26031073 0.79 RXRA (0.48) RXRAGRIN1GRIN2BNPC1RAB9A
SCHEMBL2412730 0.79 RXRA (0.42) RXRAGRIN1GRIN2BNPC1RAB9A
SCHEMBL6275209 0.78 RAB9A (0.44) RXRAGRIN1GRIN2BNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247596-A2 NOVEL PYRAZOLO [3, 4 -D] PYRIMIDINE DERIVATIVES AS ANTI -CANCER AGENTS Natco Pharma Limited (IN) 2010-11-10 EP claimed
WO-2009098715-A2 NOVEL PYRAZOLO [3, 4 -D] PYRIMIDINE DERIVATIVES AS ANTI -CANCER AGENTS NATCO PHARMA LIMITED (IN) 2009-08-13 WO claimed