SCHEMBL3424943

SCHEMBL3424943

CN1CCN(CCOc2ccc(-c3ccc4c(c3)c3c(Cl)ccnc3n4S(=O)(=O)c3ccccc3)cc2)CC1.CN1CCN(CCOc2ccc(-c3ccc4c(c3)c3ccc(Cl)nc3n4S(=O)(=O)c3ccccc3)cc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
BMP4 P12644 1/20 0.37
HTR6 P50406 4/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
KDR P35968 1/20 0.37
SRC P12931 1/20 0.36
HTR1A P08908 1/20 0.36
HTR7 P34969 1/20 0.36
LTA4H P09960 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
CXCR1 P25024 1/20 0.36
AIMP2 Q13155 1/20 0.36
EGFR P00533 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3664144 0.93 NPC1 (0.43) NPC1RAB9ABMP4HTR6KDM4E
SCHEMBL3671386 0.93 NPC1 (0.43) NPC1RAB9AHTR6KDM4EALDH1A1
SCHEMBL675636 0.81 MCHR1 (0.43) NPC1RAB9ABMP4HTR6KDM4E
SCHEMBL15375344 0.79 ALK (0.53) HTR6HTR1A
SCHEMBL3398593 0.78 LSS (0.45) HTR6KDRSRCHTR1AHTR7
SCHEMBL3398885 0.78 LSS (0.45) HTR6ALDH1A1SRCCXCR1
SCHEMBL3670674 0.78 DRD3 (0.41) HTR6KDM4EALDH1A1
SCHEMBL3672655 0.78 DRD3 (0.42) HTR6ALDH1A1
SCHEMBL677032 0.77 HTR6 (0.42) RAB9AHTR6KDM4EALDH1A1KDR
SCHEMBL675245 0.77 HTR6 (0.45) RAB9AHTR6ALDH1A1KDRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010025872-A2 ALFA-CARBOLINE INHIBITORS OF NPM-ALK, RET, AND BCR-ABL UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2010-03-11 WO disclosed