SCHEMBL3671386

SCHEMBL3671386

CN1CCN(CCOc2ccc(-c3ccc4c(c3)c3ccc(Cl)nc3n4S(=O)(=O)c3ccccc3)cc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
HTR6 P50406 4/20 0.42
KDR P35968 1/20 0.41
LTA4H P09960 2/20 0.41
HTR1A P08908 3/20 0.41
HTR7 P34969 3/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CXCR1 P25024 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
MCHR1 Q99705 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3424943 0.93 NPC1 (0.38) NPC1RAB9AHTR6KDRLTA4H
SCHEMBL675636 0.87 MCHR1 (0.43) NPC1RAB9AHTR6KDRLTA4H
SCHEMBL3664144 0.85 NPC1 (0.43) NPC1RAB9AHTR6KDRLTA4H
SCHEMBL3398885 0.84 LSS (0.45) HTR6ALDH1A1CXCR1
SCHEMBL3672655 0.83 DRD3 (0.42) HTR6ALDH1A1
SCHEMBL675245 0.82 HTR6 (0.45) RAB9AHTR6KDRALDH1A1
SCHEMBL3668236 0.81 HTR6 (0.46) HTR6
SCHEMBL675472 0.77 SRC (0.43) HTR6
SCHEMBL676293 0.77 NPC1 (0.45) NPC1RAB9AHTR6ALDH1A1
SCHEMBL677405 0.73 HTR1A (0.43) HTR6LTA4HHTR1AHTR7KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed