SCHEMBL3672655

SCHEMBL3672655

CCN(CC)CCCOc1ccc(-c2ccc3c(c2)c2ccc(Cl)nc2n3S(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 8/20 0.42
DRD2 P14416 7/20 0.42
ATP4A P20648 2/20 0.41
ATP4B P51164 2/20 0.41
HRH3 Q9Y5N1 3/20 0.41
HTR6 P50406 1/20 0.40
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PTPN1 P18031 1/20 0.39
CHEK1 O14757 1/20 0.38
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3398885 0.92 LSS (0.45) DRD3DRD2HTR6ALDH1A1TP53
SCHEMBL675362 0.86 DRD3 (0.41) DRD3DRD2ATP4AATP4BHRH3
SCHEMBL3670674 0.84 DRD3 (0.41) DRD3DRD2ATP4AATP4BHRH3
SCHEMBL675245 0.83 HTR6 (0.45) HTR6ALDH1A1TP53TSHRPSEN1
SCHEMBL3671386 0.83 NPC1 (0.43) HTR6ALDH1A1
SCHEMBL3668236 0.82 HTR6 (0.46) HTR6PSEN1PSEN2APH1BNCSTN
SCHEMBL675472 0.78 SRC (0.43) HTR6PSEN1PSEN2APH1BNCSTN
SCHEMBL3424943 0.78 NPC1 (0.38) HTR6ALDH1A1
SCHEMBL3398593 0.77 LSS (0.45) DRD3DRD2HTR6SMN1; SMN2
SCHEMBL675444 0.73 HTR6 (0.46) HTR6ALDH1A1TSHRSMN1; SMN2PSEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895744-B2 Alfa-carboline inhibitors of NPM-ALK, RET, and Bcr-Abl UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2014-11-25 US disclosed
EP-2161271-A1 Alpha-carboline inhibitors of NMP-ALK, RET, and Bcr-Abl Università Degli Studi Di Milano - Bicocca (IT) 2010-03-10 EP disclosed