SCHEMBL3425916

SCHEMBL3425916

CCc1cccc(C(N)=O)c1-c1ccc2cc[nH]c2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.45
BTK Q06187 1/20 0.45
PI4K2A Q9BTU6 1/20 0.44
PDPK1 O15530 1/20 0.43
RIPK2 O43353 1/20 0.42
JAK2 O60674 1/20 0.41
JAK3 P52333 1/20 0.41
BRD4 O60885 1/20 0.40
PARP1 P09874 3/20 0.40
MPO P05164 2/20 0.40
MAOA P21397 2/20 0.39
IKBKB O14920 3/20 0.39
CHUK O15111 3/20 0.39
PARP2 Q9UGN5 1/20 0.39
CTSL P07711 1/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3425920 0.81 LCK (0.52) LCKBTKPI4K2APDPK1RIPK2
SCHEMBL28136345 0.76 LCK (0.56) LCKBTKPI4K2APDPK1RIPK2
SCHEMBL27682000 0.76 LCK (0.56) LCKBTKPI4K2APDPK1RIPK2
SCHEMBL30369932 0.76 LCK (0.56) LCKBTKPI4K2APDPK1RIPK2
SCHEMBL11890138 0.76 TRPA1 (0.58) BTKRIPK2JAK2JAK3
SCHEMBL17500264 0.75 DHODH (0.48) LCKBTKJAK2JAK3BRD4
SCHEMBL3663816 0.73 CCNT1 (0.58) LCKBTKPI4K2ARIPK2IKBKB
SCHEMBL28555354 0.71 KDM4E (0.49) LCKBTKPI4K2ABRD4MPO
SCHEMBL4285442 0.69 NPC1 (0.45) PARP1IKBKBKDM4E
SCHEMBL23647144 0.69 PKN1 (0.47) PARP1IKBKBCHUKPARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010025872-A2 ALFA-CARBOLINE INHIBITORS OF NPM-ALK, RET, AND BCR-ABL UNIVERSITA' DEGLI STUDI DI MILANO-BICOCCA (IT) 2010-03-11 WO disclosed