SCHEMBL3428023

SCHEMBL3428023

COc1cc(F)cc(-c2cc(OC(=O)O)nn2-c2cccc(Cl)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 8/20 0.54
SLC16A1 P53985 8/20 0.54
MCTS1 Q9ULC4 2/20 0.48
PPP1CA P62136 1/20 0.44
RXRA P19793 2/20 0.43
RXRB P28702 2/20 0.43
RXRG P48443 2/20 0.43
CCKAR P32238 3/20 0.42
RPA1 P27694 3/20 0.41
NSD2 O96028 1/20 0.40
NSD1 Q96L73 1/20 0.40
NSD3 Q9BZ95 1/20 0.40
LPAR5 Q9H1C0 1/20 0.40
HPSE Q9Y251 1/20 0.40
MARS1 P56192 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3428855 0.90 PPP1CA (0.50) SLC16A3SLC16A1MCTS1PPP1CARXRA
SCHEMBL3427568 0.89 RPA1 (0.46) SLC16A3SLC16A1MCTS1RXRARXRB
SCHEMBL3429676 0.89 PPP1CA (0.46) SLC16A3SLC16A1MCTS1PPP1CARXRA
SCHEMBL3432282 0.88 RXRA (0.52) SLC16A3SLC16A1MCTS1PPP1CARXRA
SCHEMBL3428152 0.88 SLC16A3 (0.50) SLC16A3SLC16A1MCTS1PPP1CARXRA
SCHEMBL3430532 0.87 SLC16A3 (0.62) SLC16A3SLC16A1MCTS1PPP1CACCKAR
SCHEMBL1765022 0.85 PPP1CA (0.63) SLC16A3SLC16A1MCTS1PPP1CACCKAR
SCHEMBL3428061 0.83 SLC16A3 (0.48) SLC16A3SLC16A1MCTS1RPA1NSD2
SCHEMBL3434215 0.83 PGR (0.44) SLC16A3SLC16A1MCTS1PPP1CARXRA
SCHEMBL1110857 0.81 PPP1CA (0.57) SLC16A3SLC16A1MCTS1PPP1CARXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2254885-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AiCuris GmbH & Co. KG (DE) 2010-12-01 EP disclosed
WO-2009115213-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AICURIS GMBH & CO. KG (DE) 2009-09-24 WO disclosed