SCHEMBL3429299

SCHEMBL3429299

CCOC(=O)Oc1cc(-c2cccc(F)c2)n(-c2cccc(OC)c2)n1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
SLC16A3 O15427 7/20 0.44
SLC16A1 P53985 7/20 0.44
MCTS1 Q9ULC4 3/20 0.44
FAAH O00519 3/20 0.42
MAPT P10636 2/20 0.41
POLB P06746 1/20 0.41
THRB P10828 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
GAA P10253 1/20 0.40
RAB9A P51151 1/20 0.40
LMNA P02545 1/20 0.40
MGLL Q99685 1/20 0.40
TRPM8 Q7Z2W7 1/20 0.40
P2RX7 Q99572 1/20 0.40
SLC5A1 P13866 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3426584 0.88 SLC16A3 (0.57) ALDH1A1NPSR1SLC16A3SLC16A1MCTS1
SCHEMBL3431434 0.88 CHRNA7 (0.47) ALDH1A1NPSR1FAAHTHRBCA9
SCHEMBL1110815 0.87 SLC5A1 (0.47) ALDH1A1NPSR1SLC16A3SLC16A1MCTS1
SCHEMBL3428061 0.86 SLC16A3 (0.48) SLC16A3SLC16A1MCTS1MAPTPOLB
SCHEMBL3431896 0.85 FAAH (0.47) SLC16A3SLC16A1MCTS1FAAHTHRB
SCHEMBL3428152 0.85 SLC16A3 (0.50) ALDH1A1NPSR1SLC16A3SLC16A1MCTS1
SCHEMBL3427610 0.84 RPA1 (0.45) ALDH1A1FAAHPOLBTHRBMGLL
SCHEMBL1765356 0.84 FAAH (0.56) ALDH1A1NPSR1FAAHPOLBTHRB
SCHEMBL3431941 0.82 ALDH1A1 (0.45) ALDH1A1NPSR1SLC16A3SLC16A1MCTS1
SCHEMBL3431428 0.80 RXRA (0.47) ALDH1A1NPSR1SLC16A3SLC16A1MCTS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2254885-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AiCuris GmbH & Co. KG (DE) 2010-12-01 EP disclosed
WO-2009115213-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AICURIS GMBH & CO. KG (DE) 2009-09-24 WO disclosed