SCHEMBL3429446

SCHEMBL3429446

CCOC(=O)Oc1cc(-c2cccc(OCc3ccccc3)c2)n(-c2cccc(Cl)c2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 4/20 0.48
SLC16A1 P53985 4/20 0.48
MCTS1 Q9ULC4 1/20 0.48
BCHE P06276 1/20 0.46
LIPC P11150 1/20 0.46
ACHE P22303 1/20 0.46
LIPE Q05469 1/20 0.46
FAAH O00519 3/20 0.45
MDM2 Q00987 2/20 0.45
SLC5A1 P13866 3/20 0.45
MGLL Q99685 2/20 0.42
FABP3 P05413 2/20 0.42
FABP4 P15090 2/20 0.42
BCL2 P10415 1/20 0.42
MCL1 Q07820 1/20 0.42
JAK2 O60674 2/20 0.42
JAK3 P52333 1/20 0.42
JAK1 P23458 1/20 0.42
GABRA2 P47869 1/20 0.41
GABRB2 P47870 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3430971 0.89 SLC16A3 (0.50) SLC16A3SLC16A1MCTS1BCHELIPC
SCHEMBL3431644 0.88 SLC16A3 (0.46) SLC16A3SLC16A1MCTS1FAAHSLC5A1
SCHEMBL1110698 0.88 PPP1CA (0.50) SLC16A3SLC16A1MCTS1FAAHMDM2
SCHEMBL3429795 0.87 SLC16A3 (0.45) SLC16A3SLC16A1MCTS1FAAHSLC5A1
SCHEMBL3426584 0.87 SLC16A3 (0.57) SLC16A3SLC16A1MCTS1FAAHMGLL
SCHEMBL1764908 0.85 FAAH (0.59) SLC16A3SLC16A1MCTS1BCHELIPC
SCHEMBL3430158 0.85 SLC16A3 (0.43) SLC16A3SLC16A1MCTS1FAAHSLC5A1
SCHEMBL3430227 0.85 ALDH1A1 (0.45) SLC16A3SLC16A1MCTS1FAAHMGLL
SCHEMBL1110679 0.84 SLC5A1 (0.51) SLC16A3SLC16A1MCTS1FAAHSLC5A1
SCHEMBL3431968 0.82 AVPR1B (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2254885-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AiCuris GmbH & Co. KG (DE) 2010-12-01 EP disclosed
WO-2009115213-A1 (PYRAZOLYL CARBONYL)IMIDAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF RETROVIRAL DISEASES AICURIS GMBH & CO. KG (DE) 2009-09-24 WO disclosed