SCHEMBL3431340

SCHEMBL3431340

COc1cccc2c1C(c1cc3cc(N)ccc3nc1N)CC2

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.38
TLR8 Q9NR97 1/20 0.36
DRD3 P35462 1/20 0.36
PDPK1 O15530 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRA1A P35348 1/20 0.36
HTR1A P08908 6/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28789862 0.86 KDM4E (0.36) DRD2ADRA2AADRA1AHTR1A
SCHEMBL27822668 0.83 PLAU (0.31) DRD2DRD3
SCHEMBL2247023 0.82 DRD2 (0.38) DRD2TLR8DRD3HTR1A
SCHEMBL3410984 0.79 CYP19A1 (0.37) DRD2TLR8PDPK1ADRA2AADRA1A
SCHEMBL3430394 0.78 ADRA1A (0.42) ADRA2AADRA1A
SCHEMBL4109733 0.78 ADRA1A (0.42) ADRA2AADRA1A
SCHEMBL2240638 0.76 GID4 (0.37) DRD2TLR8
SCHEMBL3433618 0.75 IDO1 (0.39)
SCHEMBL3412191 0.74 HTR1A (0.42) DRD2HTR1A
SCHEMBL3432049 0.73 IDO1 (0.39) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262789-A1 2-AMINOQUINOLINES F. Hoffmann-La Roche AG (CH) 2010-12-22 EP disclosed
WO-2009109477-A1 2-AMINOQUINOLINES F. HOFFMANN-LA ROCHE AG (CH) 2009-09-11 WO disclosed