SCHEMBL3433959

SCHEMBL3433959

CS(=O)(=O)c1c(C(N)=O)ccn1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.49
MAPK1 P28482 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.40
RIPK2 O43353 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
COMT P21964 1/20 0.37
PARP1 P09874 2/20 0.36
KDM4E B2RXH2 2/20 0.36
BRD4 O60885 1/20 0.36
LMNA P02545 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
PKM P14618 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
ADORA1 P30542 1/20 0.36
KAT2B Q92831 1/20 0.36
PARP2 Q9UGN5 1/20 0.35
PARP3 Q9Y6F1 1/20 0.35
BCAT2 O15382 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28037281 0.75 NOTUM (0.51) NOTUMMAPK1SMN1; SMN2RIPK2MEN1
SCHEMBL10719764 0.72 NOTUM (0.49) NOTUMMAPK1SMN1; SMN2RIPK2MEN1
SCHEMBL8506114 0.71 ATM (0.43) NOTUMSMN1; SMN2MEN1KMT2ACOMT
SCHEMBL4783773 0.71 NOTUM (0.47) NOTUMMAPK1SMN1; SMN2RIPK2PARP1
SCHEMBL8505536 0.68 PTGS2 (0.39) NOTUMSMN1; SMN2COMTDDB1CRBN
SCHEMBL8634801 0.67 ATM (0.46) NOTUMSMN1; SMN2MEN1KMT2ACOMT
SCHEMBL1396731 0.67 MAPK1 (0.58) NOTUMMAPK1SMN1; SMN2RIPK2PARP1
SCHEMBL27944336 0.67 NOTUM (0.50) NOTUMMAPK1SMN1; SMN2MEN1KMT2A
SCHEMBL3260482 0.66 NOTUM (1.00) NOTUMMAPK1MEN1KMT2ACOMT
Hydrochloric Acid SCHEMBL29908833 0.66 MAPK1 (0.56) NOTUMMAPK1SMN1; SMN2RIPK2PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010042626-A1 1-PHENYLPYRROLE COMPOUNDS EXELIXIS, INC. (US) 2010-04-15 WO disclosed